dit workbook 2013
DESCRIPTION
2013 Workbook for STEP PrepTRANSCRIPT
Heart Rate goes downEye meiosisSalivary gland secretionBronchiolar smooth muscle CONSTRICTIONBladder wall CONSTRICTION and sphincter relaxationGU erectionGI tract motility increased and spincters relaxed
Pralidoxime regenerates Achase after organophosphate poisoning
Atropine
Donepezil, Galantine, Rivastigamine
Alzheimer’s, treat with galantine, donepezil, rivastigamine
Organophosphate poisoning, treat with atropine and pralidoxime
DUMBELSS: Diarrhea, urination, meiosis, bradycardia, bronchospasm, excitation of skeletal muscle, lacrimation, sweating, salivation
Pralidoxime
Epithelial cells?
Opposite of dumbbelss, so constipation, urinary retention, tachycardia, bronchorelaxation, loss of stimualation to skeletal muscle, dry eyes/mouth, no sweat
AntiCholinesterase
Direct Muscarinic Agonist
Muscarinic Agonist
Muscarinic Antagonist
Anticholinesterase
Acetylcholinesterase Regenerator
Cholinergic Agonist
Anticholinesterase
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Muscarinic Antagonist
Anticholinesterase
Muscarinic Antagonist
Muscarinic Antagonist
Anticholinesterase
Muscarinic Antagonist
Anticholinesterase
Cholinergic Agonist
Ipratropium, Tiotropium
Cocaine, TCA
Calcium, amphetime, ephedrine, tyramine
Cutesies have 1 M&MMAD 2s
Gq
Gi
Gs
Gs
Gq
Gi
Gq
Gi
Gs proteinAdenylcate cyclaseIncreased cAMPProtein Kinase C Activation =
Vd = D/cCL = Rate of elimination/Plasma concentrationCL = (0.7 x Vd) x T1/2LD (loading dose) = Css x VdMD (Maintenance dose) = Css x CL
10.5
600 mg
Stop the infusion for one half life which as we calculated was 10.5 h
20 mg / h
LD will not changeMD will change getting decreased