scheduling actions controlled substances...
TRANSCRIPT
U.S. Department of Justice Drug Enforcement Administration Office of Diversion Control Drug & Chemical Evaluation Section
Lists of:
Scheduling Actions
Controlled Substances
Regulated Chemicals
August 2016
Foreword The first three sections of this booklet list the names of the substances which are described in the Code of Federal
Regulations (CFR) as well as some of those which generate frequent inquiries. The substances are first arranged
alphabetically, then by Drug Enforcement Administration (DEA) drug code number, and finally by Controlled Substances
Act (21 U.S.C. §801 et seq.) (CSA) schedule.
These lists describe the basic or parent chemical and do not describe the salts, isomers, salts of isomers, esters,
ethers, and derivatives which may be controlled substances. These are not comprehensive lists so please note that a
substance need not be listed as a controlled substance to be treated as a scheduled substance for criminal prosecution.
The “Other Names” column, provides some examples of alternate names for certain compounds, and in some
instances provides examples of “positional isomers”. If outside parties want to ensure that a compound is not
considered a scheduled substance or listed chemical, they should write the DEA, Drug and Chemical Evaluation
Section (ODE), Office of Diversion Control, 8701 Morrissette Drive, Springfield, Virginia 22152, for an official
determination.
A substance (not included on these lists) may also be regulated as a controlled substance analogue. A controlled
substance analogue is a substance which is intended for human consumption, is structurally substantially similar to a schedule
I or schedule II substance, is pharmacologically substantially similar to a schedule I or schedule II substance, or is
represented as being similar to a schedule I or schedule II substance and is not an approved medication in the United States.
See 21 U.S.C. § 802(32)(A) for the definition of a controlled substance analogue and 21 U.S.C. § 813 for the schedule.
The next two sections of this booklet list the Federal Register notices through which the DEA has directed substances
to be added, deleted or transferred between schedules of the CSA. The scheduling changes are listed first in alphabetical
order by substance and then in chronological order by effective date. With the exception of anabolic steroids, section 812 of
the CSA lists only those substances which were controlled in 1970 when the law was enacted. Since then, over 200
substances have been added, removed, or transferred from one schedule to another. The current official list of controlled
substances can be found in section 1308 of the most recent issue of Title 21 Code of Federal Regulations Part 1300 to end (21
CFR § 1308) and the final rules which have been published in the Federal Register subsequent to the issuance of the CFR.
The CFR and the Federal Register are available on the U.S. Government Printing Office web site at www.gpoaccess.gov.
This information is accessible, also, on the Office of Diversion Control’s website at www.deadiversion.usdoj.gov.
The last section of this booklet identifies the “List I” and “List II” chemicals. Certain commercial transactions
involving these chemicals are regulated by the CSA. See 21 CFR §§ 1309, 1310 and 1313 for details.
These lists are intended as general references and are not comprehensive listings of all controlled substances and
regulated chemicals.
Drug and Chemical Evaluation Section Office of Diversion Control
Drug Enforcement Administration
Telephone: 202-307-7183 • FAX: 202-353-1263
August 2016
Abbreviations 2C-B = 4-Bromo-2,5-dimethoxyphenethylamine
2C-T-7 = 2,5-Dimethoxy-4(n)-propylthiophenethylamine
BZP = N-Benzylpiperazine
DMT = Dimethyltryptamine
DOM = 4-Methyl-2,5-dimethoxyamphetamine
GBL = Gamma butyrolactone
GHB = Gamma hydroxybutyric acid, gamma hydroxybutyrate, 4-hydroxybutanoic acid, sodium oxybate
LAAM = Levo-alphacetylmethadol
LSD = Lysergic acid diethylamide, lysergide
MDA = 3,4-Methylenedioxyamphetamine
MDE = 3,4-Methylenedioxy-N-ethylamphetamine
MDMA = 3,4-Methylenedioxymethamphetamine
MPPP = 1-Methyl-4-phenyl-4-propionoxypiperidine
P2P = Phenyl-2-propanone, phenylacetone
PCC = 1-Piperidinocyclohexanecarbonitrile
PCE = N-Ethyl-1-phenylcyclohexylamine
PCH = 1-Phenylcyclohexylamine
PCP = 1-(1-Phenylcyclohexyl)piperidine, phencyclidine
PEPAP = 1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine
PHP = 1-(1-Phenylcyclohexyl)pyrrolidine
SPA = (-)-1-Dimethylamino-1,2-diphenylethane
TCP = 1-[1-(2-Thienyl)cyclohexyl]piperidine
TCPy = 1-[1-(2-Thienyl)cyclohexyl]pyrrolidine
THC = Tetrahydrocannabinols
THG = Tetrahydrogestrinone
Scheduling Actions
- Alphabetical Order -
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)*
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3- 01-30-15 80 FR 5042 1/30/2015 I YL](NAPHTHALEN-1-YL)METHANONE (THJ-2201)*
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3- 05-16-13 78 FR 28735 5/16/2013 I TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLOURO-UR-144, XLR11)*
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III 3,17-dione)
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I METHOXYBENZYL) ETHANAMINE (25B-NBOMe)*
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2- 11-15-13 78 FR 68716 11/15/2013 I METHOXYBENZYL) ETHANAMINE (25C-NBOMe)*
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) 11-15-13 78 FR 68716 11/15/2013 I ETHANAMINE (25I-NBOMe)*
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C-T- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I 7)
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C-T- 09-20-02 67 FR 59163 9/20/2002 I 7) *
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C-T- 09-10-03 68 FR 53289 9/20/2003 I 7) **
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 04-12-13 78 FR 21818 4/12/2013 I (METHYLONE)
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I (METHYLONE)*
3,4-METHYLENEDIOXYPYROVALERONE (MDPV)* 10-21-11 76 FR 65371 10/21/2011 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I Narcotic
3-METHYLFENTANYL* 03-25-85 50 FR 11690 4/25/1985 I
3-METHYLFENTANYL** 04-24-86 51 FR 15474 4/25/1986 I
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 1 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
3-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
3-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE* 01-06-94 59 FR 00671 1/6/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE** 12-21-94 59 FR 65710 1/6/1995 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-07-14 79 FR 12938 3/7/2014 I MePPP)*
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4- 03-04-16 81 FR 11429 3/4/2016 I MePPP)**
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
4-METHYLAMINOREX* 10-15-87 52 FR 38225 10/15/1987 I
4-METHYLAMINOREX** 10-13-88 53 FR 40061 10/13/1988 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE)* 10-21-11 76 FR 65371 10/21/2011 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) ** 04-01-04 69 FR 17034 4/1/2004 I
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
ACETYL FENTANYL* (N-(1-PHENETHYLPIPERIDIN-4-YL)-N- 07-17-15 80 FR 42381 7/17/2015 I PHENYLACETAMIDE)
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
ACETYL-ALPHA-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ACETYL-ALPHA-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
ALFAXALONE (5α-PREGNAN-3α-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II Narcotic
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I Narcotic
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
ALPHA-ETHYLTRYPTAMINE* 03-12-93 58 FR 13533 3/12/1993 I
ALPHA-ETHYLTRYPTAMINE** 03-07-94 59 FR 10720 3/12/1994 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I Narcotic
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
ALPHA-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ALPHA-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 2 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP)* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP)** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP)* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP)** 03-04-16 81 FR 11429 3/4/2016 I
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I
AMINOREX* 09-21-92 57 FR 43399 9/21/1992 I
AMINOREX** 08-24-93 58 FR 44611 9/21/1993 I
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I Narcotic
BETA-HYDROXY-3-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXY-3-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I Expired 5/29/87
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
BETA-HYDROXYFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BETA-HYDROXYFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXYTHIOFENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
BRIVARACETAM (BRV; UCB-34714; BRIVIACT) 05-12-16 81 FR 29487 5/12/2016 V
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V Narcotic
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0 Superseded
10/97
BUTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
BUTYRYL FENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II Narcotic
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 3 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II Narcotic
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III en-17-ol, madol)
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV Narcotic
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II Narcotic
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification of CIV control
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I Narcotic
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV Narcotic
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V Narcotic
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification of CII control
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I Narcotic
ELUXADOLINE 08-11-15 11-12-15 80 FR 69861 12/17/2015 IV
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 4 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II Narcotic
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
FENFLURAMINE 05-06-97 05-06-97 5/6/1997 IV -> 0
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
FENFLURAMINE 05-15-03 68 FR 26247 5/15/2003 IV Withdrew
97 proposed
rule
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III products
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II Narcotic
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 5 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)* 05-31-85 50 FR 23118 7/1/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)** 06-17-86 51 FR 21911 7/1/1986 I
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
METHASTERONE ( 2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTAN-17BETA-OL-3-ONE)
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I
METHCATHINONE* 05-01-92 57 FR 18824 5/1/1992 I
METHCATHINONE** 04-29-93 58 FR 25934 5/1/1993 I
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I Narcotic
MPPP* 07-10-85 50 FR 28098 8/12/1985 I
MPPP** 08-11-86 51 FR 28695 8/12/1986 I
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3- 05-16-13 78 FR 28735 5/16/2013 I CARBOXAMIDE (APINACA, AKB48)*
N-(1-AMINO-3,3DIMETHYL-1-OXOBUTAN-2-YL)1- 02-05-16 81 FR 6171 2/5/2016 I (CYCLOHEXYLMETHYL)-1H-INDAZOLE-3CARBOXAMIDE (MAB-CHMINACA)*
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-10-14 79 FR 7577 2/10/2014 I 1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)*
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL- 02-05-16 81 FR 6175 2/5/2016 I 1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)**
N-(1-AMINO-3-METHYL- 01-30-15 80 FR 5042 1/30/2015 I 1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (AB-PINACA)*
N-(1-AMINO-3-METHYL-1- 01-30-15 80 FR 5042 1/30/2015 I OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL) 1H-INDAZOLE-3-CARBOXAMIDE (AB-CHMINACA)*
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 6 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDEFUBINACA)*
(AB-02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4- 02-05-16 81 FR 6175 2/5/2016 I FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDE (AB-FUBINACA)**
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
N,N-DIMETHYLAMPHETAMINE* 08-03-88 53 FR 29232 8/3/1988 I
N,N-DIMETHYLAMPHETAMINE** 08-02-89 54 FR 31815 8/2/1989 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
NAPHYRONE* 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE** 03-04-16 81 FR 11429 3/4/2016 I
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I Narcotic
PARA-FLUOROFENTANYL* 02-07-86 51 FR 4722 3/10/1986 I
PARA-FLUOROFENTANYL** 03-10-87 52 FR 7270 3/10/1987 I
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
PENTEDRONE* 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE** 03-04-16 81 FR 11429 3/4/2016 I
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 7 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
PENTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I Narcotic
PEPAP* 07-10-85 50 FR 28098 8/12/1985 I
PEPAP** 08-11-86 51 FR 28695 8/12/1986 I
PERAMPANEL [2-(2-OXO-1-PHENYL- 10-22-13 12-02-13 78 FR 72013 1/2/2014 III 5-PYRIDIN-2-YL-l ,2-DIHYDROPYRIDIN-3-YL)BENZONITRILE ]
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I Narcotic
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA- 11-23-11 07-30-12 77 FR 44456 8/29/2012 III ANDROSTANO[3,2-C]PRYAZOLE
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-10-14 79 FR 7577 2/10/2014 I CARBOXYLATE ( 5-FLUORO-PB–22; 5F–PB–22)*
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3- 02-05-16 81 FR 6175 2/5/2016 I CARBOXYLATE ( 5-FLUORO-PB–22; 5F–PB–22)**
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-10-14 79 FR 7577 2/10/2014 I (PB–22; QUPIC)*
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE 02-05-16 81 FR 6175 2/5/2016 I (PB–22; QUPIC)**
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II Narcotic
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II Narcotic
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I Narcotic
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 8 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
THENYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
THIAFENTANIL 08-26-16 81 FR 58834 8/26/2016 II
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
THIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I Narcotic
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3- 11-04-13 07-02-14 79 FR 37623 8/18/2014 IV METHOXYPHENYL)CYCLOHEXANOL)
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV
Scheduling Actions - Alphabetical Order
29-Aug-16 Page 9 of 9
Scheduling Actions
- Chronological Order -
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
METHAMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
AMPHETAMINE 05-26-71 07-07-71 36 FR 12734 7/7/1971 III -> II
FETAMIN 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
BIPHETAMINE & BIPHETAMINE-T 05-26-71 07-23-71 36 FR 13686 7/23/1971 III -> II
ESKATROL 05-26-71 08-18-71 36 FR 15744 8/18/1971 III -> II
NALOXONE HYDROCHLORIDE 08-19-71 09-29-71 36 FR 19116 9/29/1971 II -> 0
METHYLPHENIDATE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PHENMETRAZINE 09-17-71 10-28-71 36 FR 20686 10/28/1971 III -> II
PROPIRAM 01-29-72 37 FR 1468 1/29/1972 I Narcotic
BENZPHETAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CHLORPHENTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
CLORTERMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
FENFLURAMINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 IV
PHENDIMETRAZINE 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
MAZINDOL 05-09-73 06-15-73 38 FR 15719 6/15/1973 III
PHENTERMINE 05-09-73 07-06-73 38 FR 18013 7/6/1973 IV
DIETHYLPROPION 05-10-73 07-06-73 38 FR 18013 7/6/1973 IV
DROTEBANOL 07-03-73 38 FR 17717 8/6/1973 I Narcotic
2,5-DIMETHOXYAMPHETAMINE (DMA) 05-31-73 09-21-73 38 FR 26447 9/21/1973 I
4-BROMO-2,5-DIMETHOXYAMPHETAMINE 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
4-METHOXYAMPHETAMINE (PMA) 07-02-73 09-21-73 38 FR 26447 9/21/1973 I
METHAQUALONE 04-11-73 10-04-73 38 FR 27516 10/4/1973 II
AMOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
PENTOBARBITAL 05-31-75 11-13-73 38 FR 31310 11/13/1973 III -> II
SECOBARBITAL 05-31-73 11-13-73 38 FR 31310 11/13/1973 III -> II
ETORPHINE HYDROCHLORIDE 11-23-73 03-29-74 39 FR 11535 4/19/1974 I -> II Narcotic
NALOXONE 07-10-74 12-24-74 39 FR 44392 12/24/1974 II -> 0
PEMOLINE 11-07-74 01-28-75 40 FR 4150 1/28/1975 IV
MEBUTAMATE 12-13-74 01-30-75 40 FR 4418 1/30/1975 IV
CONCENTRATE OF POPPY STRAW 12-20-74 02-14-75 40 FR 6779 2/14/1975 II Narcotic
NALTREXONE 12-09-74 03-06-75 40 FR 10455 3/6/1975 II -> 0
DIFENOXIN 05-07-75 40 FR 19813 6/1/1975 I Narcotic
Scheduling Actions - Chronological Order
29-Aug-16 Page 1 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
OXAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
FLURAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
DIAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLORAZEPATE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CLONAZEPAM 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
CHLORDIAZEPOXIDE 01-27-75 06-04-75 40 FR 23998 7/2/1975 IV
MECLOQUALONE 05-29-75 07-08-75 40 FR 28611 7/10/1975 I
TCP (PCP ANALOG) 05-29-75 07-08-75 40 FR 28611 8/11/1975 I
MENRIUM 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
LIBRAX 06-05-75 11-11-75 40 FR 52609 11/28/1975 Exempted RX
APOMORPHINE 04-08-76 06-28-76 41 FR 26568 6/28/1976 II -> 0
NALBUPHINE 05-11-76 10-01-76 41 FR 43401 10/1/1976 II -> 0
DEXTRORPHAN 04-19-76 10-01-76 41 FR 43401 10/1/1976 I -> 0
PRAZEPAM 07-29-76 12-17-76 41 FR 55176 12/17/1976 IV
DEXTROPROPOXYPHENE 09-29-76 02-11-77 42 FR 8636 3/14/1977 IV
LOPERAMIDE 07-29-76 05-18-77 42 FR 25498 6/17/1977 V
LORAZEPAM 06-28-77 10-07-77 42 FR 54546 10/3/1977 IV
PHENCYCLIDINE (PCP) 12-19-77 01-25-78 43 FR 3359 2/24/1978 III -> II
PCC (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
PCH (PCP PRECURSOR) 03-20-78 05-17-78 43 FR 21324 6/16/1978 II
DIFENOXIN 1/2 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> V Narcotic
DIFENOXIN 1 MG WITH ATROPINE 06-26-78 08-28-78 43 FR 38382 9/27/1978 I -> IV Narcotic
PCE (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PHP (PCP ANALOG) 08-11-78 09-25-78 43 FR 43295 10/25/1978 I
PENTAZOCINE 09-13-78 01-10-79 44 FR 2169 2/9/1979 IV
TILIDINE 09-30-80 45 FR 64571 1/12/1980 I Narcotic
PHENYLACETONE (P2P) 12-12-79 44 FR 71822 2/11/1980 II
DEXTROPROPOXYPHENE 01-21-80 06-24-80 45 FR 42264 7/24/1980 IV Narcotic
DEXTROPROPOXYPHENE (BULK) 07-22-80 45 FR 48881 9/22/1980 IV -> II Narcotic
SPA (LEFETAMINE) 09-30-80 45 FR 64570 12/1/1980 IV
PIPRADROL 09-30-80 45 FR 64570 12/1/1980 IV
SUFENTANIL 09-30-80 45 FR 64571 12/1/1980 I Narcotic
TEMAZEPAM 01-05-81 04-07-81 45 FR 20671 4/7/1981 IV
FENETHYLLINE 05-01-81 07-21-81 46 FR 37503 8/20/1981 I
ALPHA-METHYLFENTANYL 08-05-81 09-22-81 46 FR 46799 9/22/1981 I Narcotic
Scheduling Actions - Chronological Order
29-Aug-16 Page 2 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
HALAZEPAM 04-29-81 10-29-81 46 FR 53407 10/29/1981 IV
ALPRAZOLAM 04-29-81 11-12-81 46 FR 55688 11/12/1981 IV
MAZINDOL 04-17-81 10-27-81 46 FR 52333 11/27/1981 III -> IV
N-ETHYLAMPHETAMINE 09-10-81 12-08-81 46 FR 59969 1/7/1982 I
LOPERAMIDE 07-28-82 11-03-82 47 FR 49840 11/3/1982 V -> 0
PARAHEXYL 08-05-82 11-22-82 47 FR 52432 12/22/1982 I
TRIAZOLAM 04-29-81 12-28-82 47 FR 57694 12/28/1982 IV
SUFENTANIL 03-20-84 05-25-84 49 FR 22074 5/25/1984 I -> II Narcotic
ALFENTANIL 06-25-84 49 FR 25849 8/24/1984 I Narcotic
METHAQUALONE 08-27-84 49 FR 33870 8/27/1984 II -> I
PINAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
OXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BROMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CAMAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOBAZAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOTIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
CLOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
DELORAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LORMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ETHYL LOFLAZEPATE 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NORDIAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
HALOXAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
KETAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
FLUNITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
LOPRAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
MEDAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NIMETAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
NITRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
ESTAZOLAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
TETRAZEPAM 08-01-84 10-05-84 49 FR 39307 11/5/1984 IV
BUPRENORPHINE 09-20-82 02-28-85 50 FR 8104 4/1/1985 II -> V Narcotic
3-METHYLFENTANYL* 03-25-85 50 FR 11690 4/25/1985 I
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)* 05-31-85 50 FR 23118 7/1/1985 I
PEPAP* 07-10-85 50 FR 28098 8/12/1985 I
MPPP* 07-10-85 50 FR 28098 8/12/1985 I
NALMEFENE 05-31-85 11-04-85 50 FR 45815 11/4/1985 II -> 0
Scheduling Actions - Chronological Order
29-Aug-16 Page 3 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
BETA-HYDROXYFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
ALPHA-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
3-METHYLTHIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THIOFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
BENZYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
ACETYL-ALPHA-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
THENYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I Expired 11/29/86
BETA-HYDROXY-3-METHYLFENTANYL* 10-29-85 50 FR 43698 11/29/1985 I
PARA-FLUOROFENTANYL* 02-07-86 51 FR 4722 3/10/1986 I
MIDAZOLAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
QUAZEPAM 02-07-86 03-25-86 51 FR 10190 3/25/1986 IV
3-METHYLFENTANYL** 04-24-86 51 FR 15474 4/25/1986 I
DRONABINOL PRODUCT (MARINOL) 10-18-85 05-13-86 51 FR 17476 5/13/1986 I -> II
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE)** 06-17-86 51 FR 21911 7/1/1986 I
MPPP** 08-11-86 51 FR 28695 8/12/1986 I
PEPAP** 08-11-86 51 FR 28695 8/12/1986 I
3-METHYLFENTANYL 04-24-86 09-22-86 51 FR 33592 9/22/1986 I Narcotic
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 07-27-84 10-14-86 51 FR 36552 11/13/1986 I
ACETYL-ALPHA-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
3-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
BETA-HYDROXY-3-METHYLFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I Expired 5/29/87
BETA-HYDROXYFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
THIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
ALPHA-METHYLTHIOFENTANYL** 11-26-86 51 FR 42834 11/29/1986 I
MPPP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I Narcotic
PEPAP 08-11-86 01-23-87 52 FR 2515 1/23/1987 I Narcotic
ALFENTANIL 04-17-86 01-23-87 52 FR 2516 1/23/1987 I -> II Narcotic
TILETAMINE/ZOLAZEPAM (TELAZOL) 08-11-86 01-21-87 52 FR 2221 2/20/1987 III
PARA-FLUOROFENTANYL** 03-10-87 52 FR 7270 3/10/1987 I
NABILONE 06-18-86 04-07-87 52 FR 11042 4/7/1987 II
3-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
PARA-FLUOROFENTANYL 03-10-87 05-29-87 52 FR 20070 5/29/1987 I Narcotic
THIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
ACETYL-ALPHA-METHYLFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
BETA-HYDROXYFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
Scheduling Actions - Chronological Order
29-Aug-16 Page 4 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
ALPHA-METHYLTHIOFENTANYL 11-28-86 05-29-87 52 FR 20070 5/29/1987 I Narcotic
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE* 10-15-87 52 FR 38225 10/15/1987 I
4-METHYLAMINOREX* 10-15-87 52 FR 38225 10/15/1987 I
BETA-HYDROXY-3-METHYLFENTANYL 11-28-86 01-08-88 53 FR 500 1/8/1988 I Narcotic
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 01-27-88 53 FR 2225 1/27/1988 I -> 0
MDMA (3,4-METHYLENEDIOXYMETHAMPHETAMINE) 02-22-88 53 FR 5156 3/23/1988 I
PROPYLHEXEDRINE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
PYROVALERONE 10-30-87 04-04-88 53 FR 10869 5/4/1988 V
MEFENOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENPROPOREX 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
FENCAMFAMIN 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
CATHINE 10-30-87 05-17-88 53 FR 17459 6/16/1988 IV
N,N-DIMETHYLAMPHETAMINE* 08-03-88 53 FR 29232 8/3/1988 I
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE** 10-13-88 53 FR 40061 10/13/1988 I
4-METHYLAMINOREX** 10-13-88 53 FR 40061 10/13/1988 I
CARFENTANIL 01-12-88 10-28-88 53 FR 43684 10/28/1988 II Narcotic
3,4-METHYLENEDIOXY-N-ETHYLAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
N-HYDROXY-3,4-METHYLENEDIOXYAMPHETAMINE 10-14-88 04-13-89 54 FR 14797 4/13/1989 I
4-METHYLAMINOREX 10-14-88 04-13-89 54 FR 14799 4/13/1989 I
1-[1-(2-THIENYL)CYCLOHEXYL]PYRROLIDINE 03-20-89 07-06-89 54 FR 28414 7/6/1989 I
N,N-DIMETHYLAMPHETAMINE** 08-02-89 54 FR 31815 8/2/1989 I
N,N-DIMETHYLAMPHETAMINE 08-02-89 02-02-90 55 FR 3586 2/2/1990 I
ANABOLIC STEROIDS PL 101-647 02-13-91 56 FR 5753 2/27/1991 III
GLUTETHIMIDE 07-26-90 03-21-91 56 FR 11930 3/21/1991 III -> II
PROPYLHEXEDRINE 12-03-91 56 FR 61372 12/3/1991 V -> 0
METHCATHINONE* 05-01-92 57 FR 18824 5/1/1992 I
BUTORPHANOL, THEBAINE DERIVED 04-03-92 07-14-92 57 FR 31126 7/14/1992 II->0 Superseded
10/97
AMINOREX* 09-21-92 57 FR 43399 9/21/1992 I
ZOLPIDEM 11-24-92 02-05-93 58 FR 7186 2/5/1993 IV
2,5-DIMETHOXY-4-ETHYLAMPHETAMINE (DOET) 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
CATHINONE 10-30-87 01-14-93 58 FR 4316 2/16/1993 I
ALPHA-ETHYLTRYPTAMINE* 03-12-93 58 FR 13533 3/12/1993 I
METHCATHINONE** 04-29-93 58 FR 25934 5/1/1993 I
LEVO-ALPHACETYLMETHADOL (LAAM) 04-28-93 08-18-93 58 FR 43795 8/18/1993 I -> II Narcotic
Scheduling Actions - Chronological Order
29-Aug-16 Page 5 of 9
FINAL ORDER
SUBSTANCE PROPOSAL FEDERAL *Scheduled under 21 USC 811(h) PUBLICATION PUBLICATION REGISTER EFFECTIVE CSA **Extension of temporary control DATE DATE CITATION DATE SCHEDULE
AMINOREX** 08-24-93 58 FR 44611 9/21/1993 I
METHCATHINONE 04-28-93 10-15-93 58 FR 53404 10/15/1993 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE* 01-06-94 59 FR 00671 1/6/1994 I
ALPHA-ETHYLTRYPTAMINE** 03-07-94 59 FR 10720 3/12/1994 I
AMINOREX 08-20-93 03-18-94 59 FR 12828 3/18/1994 I
ALPHA-ETHYLTRYPTAMINE 03-07-94 09-12-94 59 FR 46757 9/12/1994 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE** 12-21-94 59 FR 65710 1/6/1995 I
4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE 12-20-94 06-02-95 60 FR 28718 6/2/1995 I
REMIFENTANIL 09-16-96 11-05-96 61 FR 56893 11/5/1996 II Narcotic
FENFLURAMINE 05-06-97 05-06-97 5/6/1997 IV -> 0
BUTORPHANOL 07-10-97 10-01-97 62 FR 51370 10/31/1997 IV
SIBUTRAMINE 12-08-97 02-11-98 63 FR 6862 2/11/1998 IV
MODAFINIL 04-14-98 01-27-99 64 FR 4050 1/27/1999 IV
DRONABINOL PRODUCT (MARINOL) 11-05-98 07-02-99 64 FR 35928 7/2/1999 II -> III
KETAMINE 04-09-99 07-13-99 64 FR 37673 8/12/1999 III
ZALEPLON 05-05-99 09-15-99 64 FR 49982 9/15/1999 IV
GAMMA HYDROXYBUTYRIC ACID (GHB) PL 106-172 03-13-00 65 FR 13235 3/13/2000 I
GAMMA HYDROXYBUTYRIC ACID (GHB) FDA approved drug PL 106-172 03-13-00 65 FR 13235 3/13/2000 III products
DIHYDROETORPHINE (thebaine derivative) 11-17-00 65 FR 69442 11/17/2000 clarification of CII control
DICHLORALPHENAZONE (chloral hydrate compound) 12-11-00 08-16-01 66 FR 42943 8/16/2001 clarification of CIV control
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) * 09-20-02 67 FR 59161 9/20/2002 I
N-BENZYLPIPERAZINE (BZP) * 09-20-02 67 FR 59161 9/20/2002 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-20-02 67 FR 59163 9/20/2002 I T-7) *
BUPRENORPHINE 03-21-02 10-07-02 67 FR 62354 10/7/2002 V --> III
ALPHA-METHYLTRYPTAMINE (AMT) * 04-04-03 68 FR 16427 4/4/2003 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) * 04-04-03 68 FR 16427 4/4/2003 I
FENFLURAMINE 05-15-03 68 FR 26247 5/15/2003 IV Withdrew
97 proposed
rule
N-BENZYLPIPERAZINE (BZP) ** 09-10-03 68 FR 53289 9/20/2003 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-10-03 68 FR 53289 9/20/2003 I T-7) **
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) ** 09-10-03 68 FR 53289 9/20/2003 I
2,5-DIMETHOXY-4-(n)-PROPYLTHIOPHENETHYLAMINE (2C- 09-08-03 03-18-04 69 FR 12794 3/18/2004 I T-7)
Scheduling Actions - Chronological Order
29-Aug-16 Page 6 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
N-BENZYLPIPERAZINE (BZP) 09-08-03 03-18-04 69 FR 12794 3/18/2004 I
1-(3-TRIFLUOROMETHYLPHENYL)PIPERAZINE (TFMPP) 09-08-03 03-18-04 69 FR 12794 3/19/2004 I --> 0
ALPHA-METHYLTRYPTAMINE (AMT) ** 04-01-04 69 FR 17034 4/1/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) ** 04-01-04 69 FR 17034 4/1/2004 I
5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE (5-MeO-DIPT) 09-29-04 69 FR 58050 9/29/2004 I
ALPHA-METHYLTRYPTAMINE (AMT) 09-29-04 69 FR 58050 9/29/2004 I
ZOPICLONE 02-14-05 04-04-05 70 FR 16935 4/4/2005 IV
PREGABALIN 05-12-05 07-28-05 70 FR 43633 7/28/2005 V
ANABOLIC STEROIDS PL 108-358 12-16-05 70 FR 74653 1/17/2006 III
EMBUTRAMIDE 07-29-05 08-29-06 71 FR 51115 9/28/2006 III
LISDEXAMFETAMINE 02-22-07 05-03-07 72 FR 24532 6/4/2007 II
ORIPAVINE 09-24-07 72 FR 54208 9/24/2007 II
INDIPLON 01-31-08 01-31-08 1/31/2008 IV
LACOSAMIDE 03-10-09 05-21-09 74 FR 23789 6/22/2009 V
TAPENTADOL 02-17-09 05-21-09 74 FR 23790 6/22/2009 II
FOSPROPOFOL 07-23-09 10-06-09 74 FR 51234 11/5/2009 IV
BOLDIONE (Androsta-1,4-diene-3,17-dione) 04-25-08 12-04-09 74 FR 63603 1/4/2010 III
DESOXYMETHYLTESTOSTERONE (17a-methyl-5a-androst-2- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III en-17-ol, madol)
19-NOR-4,9(10)-ANDROSTADIENEDIONE (estra-4,9(10)-diene- 04-25-08 12-04-09 74 FR 63603 1/4/2010 III 3,17-dione)
4-ANILINO-N-PHENETHYL-4-PIPERIDINE (ANPP) 04-09-08 06-29-10 75 FR 37296 8/30/2010 II
5-METHOXY-N,N-DIMETHYLTRYPTAMINE 08-21-09 12-20-10 75 FR 79296 1/19/2011 I
CP-47,497 C8 HOMOLOGUE * 03-01-11 76 FR 11075 3/1/2011 I
CP-47,497 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-018 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-200 * 03-01-11 76 FR 11075 3/1/2011 I
JWH-073 * 03-01-11 76 FR 11075 3/1/2011 I
3,4-METHYLENEDIOXY-N-METHYLCATHINONE 10-21-11 76 FR 65371 10/21/2011 I (METHYLONE)*
3,4-METHYLENEDIOXYPYROVALERONE (MDPV)* 10-21-11 76 FR 65371 10/21/2011 I
4-METHYL-N-METHYLCATHINONE (MEPHEDRONE)* 10-21-11 76 FR 65371 10/21/2011 I
EZOGABINE 10-21-11 12-15-11 76 FR 77895 12/15/2011 V
CARISOPRODOL 11-17-09 12-12-11 76 FR 77330 1/11/2012 IV
JWH-018 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-200 ** 02-29-12 77 FR 12201 2/29/2012 I
JWH-073 ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 C8 HOMOLOGUE ** 02-29-12 77 FR 12201 2/29/2012 I
CP-47,497 ** 02-29-12 77 FR 12201 2/29/2012 I
Scheduling Actions - Chronological Order
29-Aug-16 Page 7 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
PROSTANOZOL (17 BETA-HYDROXY-5 ALPHA-ANDROSTANO[3,2-C]PRYAZOLE
11-23-11 07-30-12 77 FR 44456 8/29/2012 III
METHASTERONE ( 2 ALPHA-17 ALPHA-DIMETHYL-5 ALPHA-ANDROSTAN-17BETA-OL-3-ONE)
11-23-11 07-30-12 77 FR 44456 8/29/2012 III
3,4-METHYLENEDIOXY-N-METHYLCATHINONE (METHYLONE)
10-21-11 04-12-13 78 FR 21818 4/12/2013 I
N-(1-ADAMANTYL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (APINACA, AKB48)*
05-16-13 78 FR 28735 5/16/2013 I
[1-(5-FLUORO-PENTYL)1H-INDOL-3-YL](2,2,3,3-TETRAMETHYLCYCLOPROPYL)METHANONE(5-FLOURO-UR-144, XLR11)*
05-16-13 78 FR 28735 5/16/2013 I
(1-PENTYL-1H-INDOL-3-YL)(2,2,3,3-TETRAMETHYLCYCLOPROPYL)METHANONE (UR-144)*
05-16-13 78 FR 28735 5/16/2013 I
LORCASERIN 12-19-12 05-08-13 78 FR 26701 6/7/2013 IV
2-(4-IODO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25I-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
2-(4-CHLORO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25C-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
2-(4-BROMO-2,5-DIMETHOXYPHENYL)-N-(2-METHOXYBENZYL) ETHANAMINE (25B-NBOMe)*
11-15-13 78 FR 68716 11/15/2013 I
PERAMPANEL [2-(2-OXO-1-PHENYL-5-PYRIDIN-2-YL-l ,2-DIHYDROPYRIDIN-3-YL)BENZONITRILE ]
10-22-13 12-02-13 78 FR 72013 1/2/2014 III
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)*
02-10-14 79 FR 7577 2/10/2014 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDEFUBINACA)*
(AB-02-10-14 79 FR 7577 2/10/2014 I
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE ( 5-FLUORO-PB–22; 5F–PB–22)*
02-10-14 79 FR 7577 2/10/2014 I
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB–22; QUPIC)*
02-10-14 79 FR 7577 2/10/2014 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
PENTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP)* 03-07-14 79 FR 12938 3/7/2014 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP)* 03-07-14 79 FR 12938 3/7/2014 I
PENTEDRONE* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)* 03-07-14 79 FR 12938 3/7/2014 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4-MePPP)*
03-07-14 79 FR 12938 3/7/2014 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)* 03-07-14 79 FR 12938 3/7/2014 I
NAPHYRONE* 03-07-14 79 FR 12938 3/7/2014 I
BUTYLONE* 03-07-14 79 FR 12938 3/7/2014 I
ALFAXALONE (5α-PREGNAN-3α-OL-11,20-DIONE) 03-25-13 02-27-14 79 FR 10985 3/31/2014 IV
TRAMADOL (2-[(DIMETHYLAMINO)METHYL]-1-(3-METHOXYPHENYL)CYCLOHEXANOL)
11-04-13 07-02-14 79 FR 37623 8/18/2014 IV
SUVOREXANT 02-13-14 08-28-14 79 FR 52143 9/29/2014 IV
Scheduling Actions - Chronological Order
29-Aug-16 Page 8 of 9
SUBSTANCE
*Scheduled under 21 USC 811(h)
**Extension of temporary control
PROPOSAL
PUBLICATION
DATE PUBLICATION
DATE
FINAL
FEDERAL
REGISTER
CITATION
ORDER
EFFECTIVE
DATE
CSA
SCHEDULE
HYDROCODONE COMBINATION PRODUCTS 02-27-14 08-22-14 79 FR 49661 10/6/2014 III->II
NALOXEGEL 10-29-14 01-23-15 80 FR 3468 1/23/2015 II->0
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL) 1H-INDAZOLE-3-CARBOXAMIDE (AB-CHMINACA)*
01-30-15 80 FR 5042 1/30/2015 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (AB-PINACA)*
01-30-15 80 FR 5042 1/30/2015 I
[1-(5-FLUOROPENTYL)-1H-INDAZOL-3-YL](NAPHTHALEN-1-YL)METHANONE (THJ-2201)*
01-30-15 80 FR 5042 1/30/2015 I
ACETYL FENTANYL* (N-(1-PHENETHYLPIPERIDIN-4-YL)-N-PHENYLACETAMIDE)
07-17-15 80 FR 42381 7/17/2015 I
ELUXADOLINE 08-11-15 11-12-15 80 FR 69861 12/17/2015 IV
N-(1-AMINO-3,3DIMETHYL-1-OXOBUTAN-2-YL)1-(CYCLOHEXYLMETHYL)-1H-INDAZOLE-3CARBOXAMIDE (MAB-CHMINACA)*
02-05-16 81 FR 6171 2/5/2016 I
QUINOLIN-8-YL 1-PENTYL-1H-INDOLE-3-CARBOXYLATE (PB–22; QUPIC)**
02-05-16 81 FR 6175 2/5/2016 I
N-(1-AMINO-3,3-DIMETHYL-1-OXOBUTAN-2-YL)-1-PENTYL-1H-INDAZOLE-3-CARBOXAMIDE (ADB-PINACA)**
02-05-16 81 FR 6175 2/5/2016 I
N-(1-AMINO-3-METHYL-1-OXOBUTAN-2-YL)-1-(4-FLUOROBENZYL)-1H-INDAZOLE-3-CARBOXAMIDEFUBINACA)**
(AB-02-05-16 81 FR 6175 2/5/2016 I
QUINOLIN-8-YL 1-(5-FLUOROPENTYL)-1H-INDOLE-3-CARBOXYLATE ( 5-FLUORO-PB–22; 5F–PB–22)**
02-05-16 81 FR 6175 2/5/2016 I
ALPHA-PYRROLIDINOBUTIOPHENONE (α-PBP)** 03-04-16 81 FR 11429 3/4/2016 I
PENTEDRONE** 03-04-16 81 FR 11429 3/4/2016 I
PENTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
ALPHA-PYRROLIDINOPENTIOPHENONE (α-PVP)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-N-ETHYLCATHINONE (4-MEC)** 03-04-16 81 FR 11429 3/4/2016 I
4-METHYL-ALPHAPYRROLIDINOPROPIOPHENONE (4-MePPP)**
03-04-16 81 FR 11429 3/4/2016 I
4-FLUORO-N-METHYLCATHINONE (4-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
3-FLUORO-N-METHYLCATHINONE (3-FMC)** 03-04-16 81 FR 11429 3/4/2016 I
NAPHYRONE** 03-04-16 81 FR 11429 3/4/2016 I
BUTYLONE** 03-04-16 81 FR 11429 3/4/2016 I
BRIVARACETAM (BRV; UCB-34714; BRIVIACT) 05-12-16 81 FR 29487 5/12/2016 V
BUTYRYL FENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
BETA-HYDROXYTHIOFENTANYL* 05-12-16 81 FR 29492 5/12/2016 I
THIAFENTANIL 08-26-16 81 FR 58834 8/26/2016 II
Scheduling Actions - Chronological Order
Page 9 of 9 29-Aug-16
Controlled Substances
- Alphabetical Order -
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N
androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N
4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N
ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N
androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-androst-1-ene)
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P P)
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E ) 7509 I N 2C-E (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36 ethanamine (25B-NBOMe)
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 1 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) ethanamine (25C-NBOMe)
7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C- 7385 I N 2C-T-2 T-2 )
2-(4-Iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5 ethanamine (25I-NBOMe)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4 (Positional Isomer: 2,5-Dimethoxy-4-(2C-T-4 ) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7 (Positional Isomer: 2,5-Dimethoxy-4-7) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
3,4,5-Trimethoxyamphetamine 7390 I N TMA (Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-5), 2,4,6-Trimethoxy-amphetamine (TMA-6))
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
3-Methylfentanyl 9813 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone one)
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N
4-en-3-one)
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N
en-3-one)
4-Methoxyamphetamine 7411 I N PMA
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 2 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N
ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
5-Flouro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Flouro-UR-144, XLR-11 and XLR11 indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22 carboxylate)
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT (Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-MeO-DPT))
5-Methoxy-N-N-dimethyltryptamine 7431 I N 5-MeO-DMT (Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-MeO-DMT))
AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA 1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA 1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide)
Acetorphine 9319 I Y
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y
phenylacetamide)
Acetyl-alpha-methylfentanyl 9815 I Y
Acetyldihydrocodeine 9051 I Y Acetylcodone
Acetylmethadol 9601 I Y Methadyl acetate
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA yl)-1-pentyl-1H-indazole-3-carboxamide)
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Alfentanil 9737 II Y Alfenta
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Alpha-ethyltryptamine 7249 I N ET, Trip
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 3 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
Alpha-methyltryptamine 7432 I N AMT (Positional Isomer: N-Methyltryptamine)
Alphaprodine 9010 II Y Nisentil
alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-yl)pentan-1-one)(Positional isomers: 4-methyl-α-pyrrolidinobutiophenone (4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
Alprazolam 2882 IV N Xanax
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Aminorex 1585 I N has been sold as methamphetamine
Amobarbital 2125 II N Amytal, Tuinal
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Anileridine 9020 II Y Leritine
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48 indazole-3-carboxamide
Aprobarbital 2100 III N Alurate
Barbital 2145 IV N Veronal, Plexonal, barbitone
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Benzethidine 9606 I Y
Benzphetamine 1228 III N Didrex, Inapetyl
Benzylmorphine 9052 I Y
Betacetylmethadol 9607 I Y
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide
Betameprodine 9608 I Y
Betamethadol 9609 I Y
Betaprodine 9611 I Y
Bezitramide 9800 II Y Burgodin
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N
hydroxyandrost-4-en-3-one)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 4 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-propylpyrrolidin-1-yl] butanamide)
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-1-one) (Positional Isomers: tethylone (bk-MDEA; MDEC), dimethylone (bk-MDDMA; MDDMC))
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-phenethylpiperidin-4-yl)-N-phenylbutanamide
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb hydroxyandrost-4-en-3-one)
Camazepam 2749 IV N Albego, Limpidon, Paxor
Carfentanil 9743 II Y Wildnil
Carisoprodol 8192 IV N Soma
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine
Cathinone 1235 I N Constituent of "Khat" plant
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clobazam 2751 IV N Urbadan, Urbanyl
Clonazepam 2737 IV N Klonopin, Clonopin
Clonitazene 9612 I Y
Clorazepate 2768 IV N Tranxene
Clortermine 1647 III N Voranil
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 5 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Codeine methylbromide 9070 I Y
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Codeine-N-oxide 9053 I Y
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497 hydroxycyclohexyl-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue [(1R,3S)3-hydroxycyclohexyl-phenol)
Cyprenorphine 9054 I Y
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Delorazepam 2754 IV N
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha- 4000 III N 1-Testosterone androst-1-en-3-one)
Desomorphine 9055 I Y
Desoxymethyltestosterone 4000 III N
Dexfenfluramine 1670 IV N Redux
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Diampromide 9615 I Y
Diazepam 2765 IV N Valium, Diastat
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Diethylpropion 1610 IV N Tenuate, Tepanil
Diethylthiambutene 9616 I Y
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine (Positional Isomer: N-Methyl-N-isopropyltryptamine (MiPT))
Difenoxin 9168 I Y Lyspafen
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine 9120 II Y Didrate, Parzone
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others gm)
Dihydroetorphine 9334 II Y DHE
Dihydromorphine 9145 I Y
Dimenoxadol 9617 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 6 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y
Dimethyltryptamine 7435 I N DMT
Dioxaphetyl butyrate 9621 I Y
Diphenoxylate 9170 II Y
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as capsule as approved by FDA approved by FDA
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril androstan-3-one)
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Eluxadoline 9725 IV N VIBERZI
Embutramide 2020 III N Tributane
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Ethyl loflazepate 2758 IV N
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Ethylmethylthiambutene 9623 I Y
Ethylmorphine 9190 II Y Dionin
Ethylmorphine combination product 15 mg/du 9808 III Y
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Etonitazene 9624 I Y
Etorphine (except HCl) 9056 I Y
Etorphine HCl 9059 II Y M 99
Etoxeridine 9625 I Y
Ezogabine 2779 V N Potiga
Fencamfamin 1760 IV N Reactivan
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Fenfluramine 1670 IV N Pondimin, Ponderal
Fenproporex 1575 IV N Gacilin, Solvolip
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Fludiazepam 2759 IV N
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl 11beta,17beta-dihydroxyandrost-4-en-3-one)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 7 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Flurazepam 2767 IV N Dalmane
Formebolone (2-formyl-17alpha-methyl- 4000 III N Esiclene, Hubernol 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one)
Fospropofol 2138 IV N Lusedra
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu hydroxyandrostano[2,3-c]-furazan)
Furethidine 9626 I Y
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Glutethimide 2550 II N Doriden, Dorimide
Halazepam 2762 IV N Paxipam
Haloxazolam 2771 IV N
Heroin 9200 I Y Diacetylmorphine, diamorphine
Hydrocodone 9193 II Y dihydrocodeinone
Hydromorphinol 9301 I Y
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Hydroxypethidine 9627 I Y
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
Isomethadone 9226 II Y Isoamidone
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678 naphthoyl)indole)
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl) indole) 7081 I N JWH-081
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl) indole) 7122 I N JWH-122
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200 naphthoyl)indole)
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl) indole) 7203 I N JWH-203
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl) indole) 6250 I N JWH-250
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl) indole) 7398 I N JWH-398
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Ketobemidone 9628 I Y Cliradon
Lacosamide 2746 V N Vimpat
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Levomethorphan 9210 II Y
Levomoramide 9629 I Y
Levophenacylmorphan 9631 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 8 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Levorphanol 9220 II Y Levo-Dromoran
Lisdexamfetamine 1205 II N Vyvanse
Loprazolam 2773 IV N
Lorazepam 2885 IV N Ativan
Lorcaserin 1625 IV N Belviq
Lormetazepam 2774 IV N Noctamid
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Lysergic acid diethylamide 7315 I N LSD, lysergide
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1- 7032 I N MAB-CHMINACA and ADB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
Marihuana 7360 I N Cannabis, marijuana
Mazindol 1605 IV N Sanorex, Mazanor
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV
Mebutamate 2800 IV N Capla
Mecloqualone 2572 I N Nubarene
Medazepam 2836 IV N Nobrium
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N (Positional Isomers: 3-Methyl-methcathinone, Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Mescaline 7381 I N Constituent of "Peyote" cacti
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Assimil, Ermalone, Methybol, Tantarone androstan-3-one)
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Androviron, Proviron, Testiwop androstan-3-one)
Metazocine 9240 II Y
Methadone 9250 II Y Dolophine, Methadose, Amidone
Methadone intermediate 9254 II Y Methadone precursor
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Methandienone (17alpha-methyl-17beta- 4000 III N Dianabol, Metabolina, Nerobol, Perbolin hydroxyandrost-1,4-diene-3-one)
Methandriol (17alpha-methyl-3beta,17beta- 4000 III N Sinesex, Stenediol, Troformone dihydroxyandrost-5-ene)
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 9 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Methasterone (2alpha,17alpha-dimethyl-5alpha-androstan-17beta-ol-3-one)
4000 III N Methasterone
Methcathinone 1237 I N N-Methylcathinone, "cat"
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst-1-en-3-one)
4000 III N Primobolan, Primobolan Depot, Primobolan S
Methohexital 2264 IV N Brevital
Methyldesorphine 9302 I Y
Methyldienolone (17alpha-methyl-17beta-hydroxyestr-4,9(10)-dien-3-one)
4000 III N
Methyldihydromorphine 9304 I Y
Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N Methylone
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Methyltestosterone (17alpha-methyl-17beta-hydroxyandrost-4-en-3-one)
4000 III N Android, Oreton, Testred, Virilon
Methyltrienolone (17alpha-methyl-17beta-hydroxyestr-4,9,11-trien-3-one)
4000 III N Metribolone
Methyprylon 2575 III N Noludar
Metopon 9260 II Y
Mibolerone (7alpha,17alpha-dimethyl-17beta-hydroxyestr-4-en-3-one)
4000 III N Cheque, Matenon
Midazolam 2884 IV N Versed
Modafinil 1680 IV N Provigil
Moramide-intermediate 9802 II Y
Morpheridine 9632 I Y
Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR
Morphine combination product/50 mg/(100 ml or 100 gm)
9810 III Y
Morphine methylbromide 9305 I Y
Morphine methylsulfonate 9306 I Y
Morphine-N-oxide 9307 I Y
Myrophine 9308 I Y
N,N-Dimethylamphetamine 1480 I N
Nabilone 7379 II N Cesamet
Nalorphine 9400 III Y Nalline
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-(pyrrolidin-1-yl)pentan-1-one) (Positional Isomer: α-naphyrone)
N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 10 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Ethylamphetamine 1475 I N NEA
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
Nicocodeine 9309 I Y
Nicomorphine 9312 I Y Vilan
Nimetazepam 2837 IV N Erimin
Nitrazepam 2834 IV N Mogadon
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
Noracymethadol 9633 I Y
Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar en-3-one)
Norlevorphanol 9634 I Y
Normethadone 9635 I Y Phenyldimazone
Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron hydroxyestr-4-en-3-one)
Normorphine 9313 I Y
Norpipanone 9636 I Y
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Opium extracts 9610 II Y
Opium fluid extract 9620 II Y
Opium poppy 9650 II Y Papaver somniferum
Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Opium tincture 9630 II Y Laudanum
Opium, granulated 9640 II Y Granulated opium
Opium, powdered 9639 II Y Powdered opium
Opium, raw 9600 II Y Raw opium, gum opium
Oripavine 9330 II Y
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome 5alpha-androstan-3-one)
Oxazepam 2835 IV N Serax, Serenid-D
Oxazolam 2839 IV N Serenal, Convertal
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10 dihydroxyandrost-4-en-3-one)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 11 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Oxymetholone (17alpha-methyl-2-hydroxymethylene-17beta-hydroxy-5alpha-androstan-3-one)
4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd
Oxymorphone 9652 II Y Numorphan
Para-Fluorofentanyl 9812 I Y China White, fentanyl
Parahexyl 7374 I N Synhexyl,
Paraldehyde 2585 IV N Paral
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
Pemoline 1530 IV N Cylert
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone (3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
Pentobarbital 2270 II N Nembutal
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)pentan-1-one) (Positional Isomer: dibutylone (bk-DMBDB))
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Peyote 7415 I N Cactus which contains mescaline
Phenadoxone 9637 I Y
Phenampromide 9638 I Y
Phenazocine 9715 II Y Narphen, Prinadol
Phencyclidine 7471 II N PCP, Sernylan
Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Phenmetrazine 1631 II N Preludin
Phenobarbital 2285 IV N Luminal, Bellergal-S
Phenomorphan 9647 I Y
Phenoperidine 9641 I Y Operidine, Lealgin
Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Piminodine 9730 II Y
Pinazepam 2883 IV N Domar
Pipradrol 1750 IV N Detaril, Stimolag Fortis
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 12 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Piritramide 9642 I Y Piridolan
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS
Prazepam 2764 IV N Centrax
Pregabalin 2782 V N Lyrica
Proheptazine 9643 I Y
Properidine 9644 I Y
Propiram 9649 I Y Algeril
Prostanozol (17beta-hydroxy-5alpha-androstano[3,2-c]pyrazole)
4000
Psilocybin 7437
III
I
N
N
Prostanozol
Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"
Pyrovalerone 1485 V N Centroton, Thymergix
Quazepam 2881 IV N Doral
Racemethorphan 9732 II Y
Racemoramide 9645 I Y
Racemorphan 9733 II Y Dromoran
Remifentanil 9739 II Y Ultiva
Secobarbital 2315 II N Seconal, Tuinal
Secobarbital & noncontrolled active ingred 2316 III N
Secobarbital suppository dosage form 2316 III N
Sibutramine 1675 IV N Meridia
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
SR-18 (Also known as RCS-8) (1-Cyclohexylethyl-3-(2-methoxyphenylacetyl) indole)
7008
SR-19 (Also known as RCS-4) (1-Pentyl-3-[(4-methoxy)-benzoyl] indole
7104
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha-androst-2-eno[3,2-c]-pyrazole)
4000
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst-1-en-3-one)
4000
Stimulant compounds previously excepted 1405
I
I
III
III
III
N
N
N
N
N
SR-18 and RCS-8
SR-19 and RCS-4
Winstrol, Winstrol-V
Mediatric
Sufentanil 9740 II Y Sufenta
Sulfondiethylmethane 2600 III N
Sulfonethylmethane 2605 III N
Sulfonmethane 2610 III N
Suvorexant 2223
Talbutal 2100
IV
III
N
N
MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone
Lotusate
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 13 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Tapentadol 9780 II Y
Temazepam 2925 IV N Restoril
Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta- 4000 III N Teolit, Teslac 1,4-dien-17-oic acid lactone)
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and others
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta- 4000 III N THG hydroxygon-4,9,11-trien-3-one)
Tetrazepam 2886 IV N Myolastan, Musaril
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Thebaine 9333 II Y Precursor of many narcotics
Thiafentanil 9729 II Y Thianil
Thiamylal 2100 III N Surital
Thiofentanyl 9835 I Y Chine white, fentanyl
Thiopental 2100 III N Pentothal
THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3- 7024 I N THJ-2201 yl](naphthalen-1-yl)methanone
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol methoxyphenyl)cyclohexanol)
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
Triazolam 2887 IV N Halcion
Trimeperidine 9646 I Y Promedolum
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- 7144 I N UR-144 tetramethylcyclopropyl)methanone
Vinbarbital 2100 III N Delvinal, vinbarbitone
Zaleplon 2781 IV N Sonata
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - Alphabetical Order
29-Aug-16 Page 14 of 14
Controlled Substances
- by DEA Drug Code Number -
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others gm)
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Lisdexamfetamine 1205 II N Vyvanse
Benzphetamine 1228 III N Didrex, Inapetyl
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine
3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
Cathinone 1235 I N Constituent of "Khat" plant
Methcathinone 1237 I N N-Methylcathinone, "cat"
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone (3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N (Positional Isomers: 3-Methyl-methcathinone, Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-(pyrrolidin-1-yl)pentan-1-one) (Positional Isomer: α-naphyrone)
Stimulant compounds previously excepted 1405 III N Mediatric
N-Ethylamphetamine 1475 I N NEA
N,N-Dimethylamphetamine 1480 I N
Pyrovalerone 1485 V N Centroton, Thymergix
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Pemoline 1530 IV N Cylert
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 1 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Fenproporex 1575 IV N Gacilin, Solvolip
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Aminorex 1585 I N has been sold as methamphetamine
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
Mazindol 1605 IV N Sanorex, Mazanor
Diethylpropion 1610 IV N Tenuate, Tepanil
Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Lorcaserin 1625 IV N Belviq
Phenmetrazine 1631 II N Preludin
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clortermine 1647 III N Voranil
Dexfenfluramine 1670 IV N Redux
Fenfluramine 1670 IV N Pondimin, Ponderal
Sibutramine 1675 IV N Meridia
Modafinil 1680 IV N Provigil
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Pipradrol 1750 IV N Detaril, Stimolag Fortis
Fencamfamin 1760 IV N Reactivan
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Embutramide 2020 III N Tributane
Aprobarbital 2100 III N Alurate
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Talbutal 2100 III N Lotusate
Thiamylal 2100 III N Surital
Thiopental 2100 III N Pentothal
Vinbarbital 2100 III N Delvinal, vinbarbitone
Amobarbital 2125 II N Amytal, Tuinal
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Fospropofol 2138 IV N Lusedra
Barbital 2145 IV N Veronal, Plexonal, barbitone
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 2 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Suvorexant 2223 IV N MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Methohexital 2264 IV N Brevital
Pentobarbital 2270 II N Nembutal
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Phenobarbital 2285 IV N Luminal, Bellergal-S
Secobarbital 2315 II N Seconal, Tuinal
Secobarbital & noncontrolled active ingred 2316 III N
Secobarbital suppository dosage form 2316 III N
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Glutethimide 2550 II N Doriden, Dorimide
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Mecloqualone 2572 I N Nubarene
Methyprylon 2575 III N Noludar
Paraldehyde 2585 IV N Paral
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Sulfondiethylmethane 2600 III N
Sulfonethylmethane 2605 III N
Sulfonmethane 2610 III N
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-propylpyrrolidin-1-yl] butanamide)
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Clonazepam 2737 IV N Klonopin, Clonopin
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Lacosamide 2746 V N Vimpat
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Camazepam 2749 IV N Albego, Limpidon, Paxor
Clobazam 2751 IV N Urbadan, Urbanyl
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 3 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Delorazepam 2754 IV N
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Ethyl loflazepate 2758 IV N
Fludiazepam 2759 IV N
Halazepam 2762 IV N Paxipam
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Prazepam 2764 IV N Centrax
Diazepam 2765 IV N Valium, Diastat
Flurazepam 2767 IV N Dalmane
Clorazepate 2768 IV N Tranxene
Haloxazolam 2771 IV N
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Loprazolam 2773 IV N
Lormetazepam 2774 IV N Noctamid
Ezogabine 2779 V N Potiga
Zaleplon 2781 IV N Sonata
Pregabalin 2782 V N Lyrica
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta
Mebutamate 2800 IV N Capla
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Nitrazepam 2834 IV N Mogadon
Oxazepam 2835 IV N Serax, Serenid-D
Medazepam 2836 IV N Nobrium
Nimetazepam 2837 IV N Erimin
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Oxazolam 2839 IV N Serenal, Convertal
Quazepam 2881 IV N Doral
Alprazolam 2882 IV N Xanax
Pinazepam 2883 IV N Domar
Midazolam 2884 IV N Versed
Lorazepam 2885 IV N Ativan
Tetrazepam 2886 IV N Myolastan, Musaril
Triazolam 2887 IV N Halcion
Temazepam 2925 IV N Restoril
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 4 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N 4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N ene; 3alpha,17beta-dihydroxyestr-5-ene)
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-androst-1-ene)
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone one)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N 4-en-3-one)
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N en-3-one)
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb hydroxyandrost-4-en-3-one)
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Dehydrochloromethyltestosterone (4-chloro-17beta- 4000 III N Oral-Turinabol hydroxy-17alpha-methylandrost-1,4-dien-3-one)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 5 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha-androst-1-en-3-one)
4000 III N 1-Testosterone
Desoxymethyltestosterone 4000 III N
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha- 4000 III N Drolban, Masterid, Permastril androstan-3-one)
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Fluoxymesterone (9-fluoro-17alpha-methyl- 4000 III N Anadroid-F, Halotestin, Ora-Testryl 11beta,17beta-dihydroxyandrost-4-en-3-one)
Formebolone (2-formyl-17alpha-methyl- 4000 III N Esiclene, Hubernol 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one)
Furazabol (17alpha-methyl-17beta- 4000 III N Frazalon, Miotolon, Qu Zhi Shu hydroxyandrostano[2,3-c]-furazan)
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Assimil, Ermalone, Methybol, Tantarone androstan-3-one)
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Androviron, Proviron, Testiwop androstan-3-one)
Methandienone (17alpha-methyl-17beta- 4000 III N Dianabol, Metabolina, Nerobol, Perbolin hydroxyandrost-1,4-diene-3-one)
Methandriol (17alpha-methyl-3beta,17beta- 4000 III N Sinesex, Stenediol, Troformone dihydroxyandrost-5-ene)
Methasterone (2alpha,17alpha-dimethyl-5alpha- 4000 III N Methasterone androstan-17beta-ol-3-one)
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst- 4000 III N Primobolan, Primobolan Depot, Primobolan S 1-en-3-one)
Methyldienolone (17alpha-methyl-17beta-hydroxyestr- 4000 III N 4,9(10)-dien-3-one)
Methyltestosterone (17alpha-methyl-17beta- 4000 III N Android, Oreton, Testred, Virilon hydroxyandrost-4-en-3-one)
Methyltrienolone (17alpha-methyl-17beta-hydroxyestr- 4000 III N Metribolone 4,9,11-trien-3-one)
Mibolerone (7alpha,17alpha-dimethyl-17beta- 4000 III N Cheque, Matenon hydroxyestr-4-en-3-one)
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar en-3-one)
Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron hydroxyestr-4-en-3-one)
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome 5alpha-androstan-3-one)
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10 dihydroxyandrost-4-en-3-one)
Oxymetholone (17alpha-methyl-2-hydroxymethylene- 4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd 17beta-hydroxy-5alpha-androstan-3-one)
Prostanozol (17beta-hydroxy-5alpha-androstano[3,2- 4000 III N Prostanozol c]pyrazole)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 6 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha-androst-2-eno[3,2-c]-pyrazole)
4000 III N Winstrol, Winstrol-V
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst-1-en-3-one)
4000 III N
Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta-1,4-dien-17-oic acid lactone)
4000 III N Teolit, Teslac
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta-hydroxygon-4,9,11-trien-3-one)
4000 III N THG
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl) indole) 6250 I N JWH-250
SR-18 (Also known as RCS-8) (1-Cyclohexylethyl-3-(2-methoxyphenylacetyl) indole)
7008 I N SR-18 and RCS-8
5-Flouro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
7011 I N 5-Flouro-UR-144, XLR-11 and XLR11
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
7012 I N AB-FUBINACA
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
AB-PINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide)
7023 I N AB-PINACA
THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3-yl](naphthalen-1-yl)methanone
7024 I N THJ-2201
AB-CHMINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide
7031 I N AB-CHMINACA
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1-oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
7032 I N MAB-CHMINACA and ADB-CHMINACA
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide)
7035 I N ADB-PINACA
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H-indazole-3-carboxamide
7048 I N APINACA and AKB48
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl) indole) 7081 I N JWH-081
SR-19 (Also known as RCS-4) (1-Pentyl-3-[(4-methoxy)-benzoyl] indole
7104 I N SR-19 and RCS-4
JWH-018 (also known as AM678) (1-Pentyl-3-(1-naphthoyl)indole)
7118 I N JWH-018 and AM-678
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl) indole) 7122 I N JWH-122
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone
7144 I N UR-144
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1-naphthoyl)indole)
7200 I N JWH-200
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl) indole) 7203 I N JWH-203
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 7 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22 carboxylate)
Alpha-ethyltryptamine 7249 I N ET, Trip
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497 hydroxycyclohexyl-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue [(1R,3S)3-hydroxycyclohexyl-phenol)
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Lysergic acid diethylamide 7315 I N LSD, lysergide
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7 (Positional Isomer: 2,5-Dimethoxy-4-7) ethylthioamphetamine (Aleph-2))
Marihuana 7360 I N Cannabis, marijuana
Dronabinol (synthetic) in sesame oil in soft gelatin 7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as capsule as approved by FDA approved by FDA
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and others
Parahexyl 7374 I N Synhexyl,
Nabilone 7379 II N Cesamet
Mescaline 7381 I N Constituent of "Peyote" cacti
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C- 7385 I N 2C-T-2 T-2 )
3,4,5-Trimethoxyamphetamine 7390 I N TMA (Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-5), 2,4,6-Trimethoxy-amphetamine (TMA-6))
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl) indole) 7398 I N JWH-398
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
4-Methoxyamphetamine 7411 I N PMA
Peyote 7415 I N Cactus which contains mescaline
5-Methoxy-N-N-dimethyltryptamine 7431 I N 5-MeO-DMT (Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-MeO-DMT))
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 8 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Alpha-methyltryptamine 7432 I N AMT (Positional Isomer: N-Methyltryptamine)
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine (Positional Isomer: N-Methyl-N-isopropyltryptamine (MiPT))
Dimethyltryptamine 7435 I N DMT
Psilocybin 7437 I N Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT (Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-MeO-DPT))
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
Phencyclidine 7471 II N PCP, Sernylan
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E ) 7509 I N 2C-E (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-Iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P P)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4 (Positional Isomer: 2,5-Dimethoxy-4-(2C-T-4 ) ethylthioamphetamine (Aleph-2))
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36 ethanamine (25B-NBOMe)
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82 ethanamine (25C-NBOMe)
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5 ethanamine (25I-NBOMe)
Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N Methylone
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-1-one) (Positional Isomers: tethylone (bk-MDEA; MDEC), dimethylone (bk-MDDMA; MDDMC))
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 9 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)pentan-1-one) (Positional Isomer: dibutylone (bk-DMBDB))
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-yl)pentan-1-one)(Positional isomers: 4-methyl-α-pyrrolidinobutiophenone (4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Carisoprodol 8192 IV N Soma
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
Alphaprodine 9010 II Y Nisentil
Anileridine 9020 II Y Leritine
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Acetyldihydrocodeine 9051 I Y Acetylcodone
Benzylmorphine 9052 I Y
Codeine-N-oxide 9053 I Y
Cyprenorphine 9054 I Y
Desomorphine 9055 I Y
Etorphine (except HCl) 9056 I Y
Etorphine HCl 9059 II Y M 99
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Codeine methylbromide 9070 I Y
Dihydrocodeine 9120 II Y Didrate, Parzone
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Dihydromorphine 9145 I Y
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Difenoxin 9168 I Y Lyspafen
Diphenoxylate 9170 II Y
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Ethylmorphine 9190 II Y Dionin
Hydrocodone 9193 II Y dihydrocodeinone
Heroin 9200 I Y Diacetylmorphine, diamorphine
Levomethorphan 9210 II Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 10 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Levorphanol 9220 II Y Levo-Dromoran
Isomethadone 9226 II Y Isoamidone
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Metazocine 9240 II Y
Methadone 9250 II Y Dolophine, Methadose, Amidone
Methadone intermediate 9254 II Y Methadone precursor
Metopon 9260 II Y
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR
Hydromorphinol 9301 I Y
Methyldesorphine 9302 I Y
Methyldihydromorphine 9304 I Y
Morphine methylbromide 9305 I Y
Morphine methylsulfonate 9306 I Y
Morphine-N-oxide 9307 I Y
Myrophine 9308 I Y
Nicocodeine 9309 I Y
Nicomorphine 9312 I Y Vilan
Normorphine 9313 I Y
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Acetorphine 9319 I Y
Oripavine 9330 II Y
Thebaine 9333 II Y Precursor of many narcotics
Dihydroetorphine 9334 II Y DHE
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Nalorphine 9400 III Y Nalline
Opium, raw 9600 II Y Raw opium, gum opium
Acetylmethadol 9601 I Y Methadyl acetate
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 11 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Benzethidine 9606 I Y
Betacetylmethadol 9607 I Y
Betameprodine 9608 I Y
Betamethadol 9609 I Y
Opium extracts 9610 II Y
Betaprodine 9611 I Y
Clonitazene 9612 I Y
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Diampromide 9615 I Y
Diethylthiambutene 9616 I Y
Dimenoxadol 9617 I Y
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y
Opium fluid extract 9620 II Y
Dioxaphetyl butyrate 9621 I Y
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Ethylmethylthiambutene 9623 I Y
Etonitazene 9624 I Y
Etoxeridine 9625 I Y
Furethidine 9626 I Y
Hydroxypethidine 9627 I Y
Ketobemidone 9628 I Y Cliradon
Levomoramide 9629 I Y
Opium tincture 9630 II Y Laudanum
Levophenacylmorphan 9631 I Y
Morpheridine 9632 I Y
Noracymethadol 9633 I Y
Norlevorphanol 9634 I Y
Normethadone 9635 I Y Phenyldimazone
Norpipanone 9636 I Y
Phenadoxone 9637 I Y
Phenampromide 9638 I Y
Opium, powdered 9639 II Y Powdered opium
Opium, granulated 9640 II Y Granulated opium
Phenoperidine 9641 I Y Operidine, Lealgin
Piritramide 9642 I Y Piridolan
Proheptazine 9643 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 12 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Properidine 9644 I Y
Racemoramide 9645 I Y
Trimeperidine 9646 I Y Promedolum
Phenomorphan 9647 I Y
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Propiram 9649 I Y Algeril
Opium poppy 9650 II Y Papaver somniferum
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Oxymorphone 9652 II Y Numorphan
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Phenazocine 9715 II Y Narphen, Prinadol
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Eluxadoline 9725 IV N VIBERZI
Thiafentanil 9729 II Y Thianil
Piminodine 9730 II Y
Racemethorphan 9732 II Y
Racemorphan 9733 II Y Dromoran
Alfentanil 9737 II Y Alfenta
Remifentanil 9739 II Y Ultiva
Sufentanil 9740 II Y Sufenta
Carfentanil 9743 II Y Wildnil
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol methoxyphenyl)cyclohexanol)
Tapentadol 9780 II Y
Bezitramide 9800 II Y Burgodin
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Moramide-intermediate 9802 II Y
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Ethylmorphine combination product 15 mg/du 9808 III Y
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Morphine combination product/50 mg/(100 ml or 100 9810 III Y gm)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 13 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Para-Fluorofentanyl 9812 I Y China White, fentanyl
3-Methylfentanyl 9813 I Y China White, fentanyl
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Acetyl-alpha-methylfentanyl 9815 I Y
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y phenylacetamide)
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-phenethylpiperidin-4-yl)-N-phenylbutanamide
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
Thiofentanyl 9835 I Y Chine white, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by DEA Drug Code Number
29-Aug-16 Page 14 of 14
Controlled Substances
- by CSA Schedule -
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
1-(1-Phenylcyclohexyl)pyrrolidine 7458 I N PCPy, PHP, rolicyclidine
1-(2-Phenylethyl)-4-phenyl-4-acetoxypiperidine 9663 I Y PEPAP, synthetic heroin
1-[1-(2-Thienyl)cyclohexyl]piperidine 7470 I N TCP, tenocyclidine
1-[1-(2-Thienyl)cyclohexyl]pyrrolidine 7473 I N TCPy
1-Methyl-4-phenyl-4-propionoxypiperidine 9661 I Y MPPP, synthetic heroin
2-(2,5-Dimethoxy-4-(n)-propylphenyl) ethanamine (2C- 7524 I N 2C-P P)
2-(2,5-Dimethoxy-4-ethylphenyl) ethanamine (2C-E ) 7509 I N 2C-E (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
2-(2,5-Dimethoxy-4-methylphenyl) ethanamine (2C-D) 7508 I N 2C-D
2-(2,5-Dimethoxy-4-nitro-phenyl) ethanamine (2C-N) 7521 I N 2C-N
2-(2,5-Dimethoxyphenyl) ethanamine (2C-H) 7517 I N 2C-H
2-(4-bromo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7536 I N 25B-NBOMe, 2C-B-NBOMe, 25B, Cimbi-36 ethanamine (25B-NBOMe)
2-(4-Chloro-2,5-dimethoxyphenyl) ethanamine (2C-C) 7519 I N 2C-C
2-(4-chloro-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7537 I N 25C-NBOMe, 2C-C-NBOMe, 25C, Cimbi-82 ethanamine (25C-NBOMe)
2-(4-Ethylthio-2,5-dimethoxyphenyl) ethanamine (2C- 7385 I N 2C-T-2 T-2 )
2-(4-Iodo-2,5-dimethoxyphenyl) ethanamine (2C-I) 7518 I N 2C-I
2-(4-iodo-2,5-dimethoxyphenyl)-N-(2-methoxybenzyl) 7538 I N 25I-NBOMe, 2C-I-NBOMe, 25I, Cimbi-5 ethanamine (25I-NBOMe)
2-(4-Isopropylthio)-2,5-dimethoxyphenyl) ethanamine 7532 I N 2C-T-4 (Positional Isomer: 2,5-Dimethoxy-4-(2C-T-4 ) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-(n)-propylthiophenethylamine (2C-T- 7348 I N 2C-T-7 (Positional Isomer: 2,5-Dimethoxy-4-7) ethylthioamphetamine (Aleph-2))
2,5-Dimethoxy-4-ethylamphetamine 7399 I N DOET
2,5-Dimethoxyamphetamine 7396 I N DMA, 2,5-DMA
3,4,5-Trimethoxyamphetamine 7390 I N TMA (Positional Isomers: 2,4,5-Trimethoxy-amphetamine (TMA-5), 2,4,6-Trimethoxy-amphetamine (TMA-6))
3,4-Methylenedioxyamphetamine 7400 I N MDA, Love Drug
3,4-Methylenedioxymethamphetamine 7405 I N MDMA, Ecstasy, XTC
3,4-Methylenedioxy-N-ethylamphetamine 7404 I N N-ethyl MDA, MDE, MDEA
3-Fluoro-N-methylcathinone (3-FMC) 1233 I N 1-(3-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
3-Methylfentanyl 9813 I Y China White, fentanyl
3-Methylthiofentanyl 9833 I Y China White, fentanyl
4-Bromo-2,5-dimethoxyamphetamine 7391 I N DOB, 4-bromo-DMA
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 1 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
4-Bromo-2,5-dimethoxyphenethylamine 7392 I N 2C-B, Nexus, has been sold as Ecstasy, i.e. MDMA
4-Fluoro-N-methylcathinone (4-FMC) 1238 I N flephedrone; 1-(4-fluorophenyl)-2-(methylamino)propan-1-one) (Positional isomer: 2-FMC)
4-Methoxyamphetamine 7411 I N PMA
4-Methyl-2,5-dimethoxyamphetamine 7395 I N DOM, STP (Positional Isomer: 2,5-Dimethoxy-3,4-dimethylphenethylamine (2C-G))
4-Methyl-alphapyrrolidinopropiophenone (4-MePPP) 7498 I N MePPP, 4-methyl-α-pyrrolidinopropiophenone, 1-(4-methylphenyl)-2-(pyrrolidin-1-yl)-propan-1-one)
4-Methylaminorex (cis isomer) 1590 I N U4Euh, McN-422
4-Methyl-N-ethylcathinone (4-MEC) 1249 I N 2-(ethylamino)-1-(4-methylphenyl)propan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone(3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
5-Flouro-UR-144 and XLR11 [1-(5-Fluoro-pentyl)1H- 7011 I N 5-Flouro-UR-144, XLR-11 and XLR11 indol-3-yl](2,2,3,3-tetramethylcyclopropyl)methanone
5F-PB-22 (Quinolin-8-yl 1-(5-fluoropentyl)-1H-indole-3- 7225 I N 5-Fluoro-PB-22; 5F-PB-22 carboxylate)
5-Methoxy-3,4-methylenedioxyamphetamine 7401 I N MMDA
5-Methoxy-N,N-diisopropyltryptamine 7439 I N 5-MeO-DIPT (Positional Isomer: 5-Methoxy-N,N-dipropyltryptamine (5-MeO-DPT))
5-Methoxy-N-N-dimethyltryptamine 7431 I N 5-MeO-DMT (Positional Isomer: 4-Methoxy-N,N-dimethyltryptamine (4-MeO-DMT))
AB-CHMINACA (N-(1-amino-3-methyl-1- 7031 I N AB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide
AB-FUBINACA (N-(1-amino-3-methyl-1-oxobutan-2-yl)- 7012 I N AB-FUBINACA 1-(4-fluorobenzyl)-1H-indazole-3-carboxamide)
AB-PINACA (N-(1-amino-3-methyl- 7023 I N AB-PINACA 1-oxobutan-2-yl)-1-pentyl-1H-indazole-3-carboxamide)
Acetorphine 9319 I Y
Acetyl Fentanyl (N-(1-phenethylpiperidin-4-yl)-N- 9821 I Y phenylacetamide)
Acetyl-alpha-methylfentanyl 9815 I Y
Acetyldihydrocodeine 9051 I Y Acetylcodone
Acetylmethadol 9601 I Y Methadyl acetate
ADB-PINACA (N-(1-amino-3,3-dimethyl-1-oxobutan-2- 7035 I N ADB-PINACA yl)-1-pentyl-1H-indazole-3-carboxamide)
Allylprodine 9602 I Y
Alphacetylmethadol except levo-alphacetylmethadol 9603 I Y
Alpha-ethyltryptamine 7249 I N ET, Trip
Alphameprodine 9604 I Y
Alphamethadol 9605 I Y
Alpha-methylfentanyl 9814 I Y China White, fentanyl
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 2 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Alpha-methylthiofentanyl 9832 I Y China White, fentanyl
Alpha-methyltryptamine 7432 I N AMT (Positional Isomer: N-Methyltryptamine)
alpha-pyrrolidinobutiophenone (α-PBP) 7546 I N 1-phenyl-2-(pyrrolidin-1-yl)butan-1-one)
alpha-pyrrolidinopentiophenone (α-PVP) 7545 I N α-pyrrolidinovalerophenone, 1-phenyl-2- (pyrrolidin-1-yl)pentan-1-one)(Positional isomers: 4-methyl-α-pyrrolidinobutiophenone (4-MePBP), 1-phenyl-2-(piperidin-1-yl)butan-1-one)
AM2201 (1-(5-Fluoropentyl)-3-(1-naphthoyl) indole) 7201 I N AM2201
AM-694 (1-(5-Fluoropentyl)-3-(2-iodobenzoyl) indole) 7694 I N AM-694
Aminorex 1585 I N has been sold as methamphetamine
APINACA and AKB48 N-(1-Adamantyl)-1-pentyl-1H- 7048 I N APINACA and AKB48 indazole-3-carboxamide
Benzethidine 9606 I Y
Benzylmorphine 9052 I Y
Betacetylmethadol 9607 I Y
Beta-hydroxy-3-methylfentanyl 9831 I Y China White, fentanyl
Beta-hydroxyfentanyl 9830 I Y China White, fentanyl
Beta-hydroxythiofentanyl 9836 I Y N-[1-[2-hydroxy-2-(thiophen-2-yl)ethyl]piperidin-4-yl]-N-phenylpropionamide, N-[1-[2-hydroxy-2-(2-thienyl)ethyl]-4-piperidinyl]-N-phenylpropanamide
Betameprodine 9608 I Y
Betamethadol 9609 I Y
Betaprodine 9611 I Y
Bufotenine 7433 I N Mappine, N,N-dimethylserotonin
Butylone 7541 I N bk-MBDB; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)butan-1-one) (Positional Isomers: tethylone (bk-MDEA; MDEC), dimethylone (bk-MDDMA; MDDMC))
Butyryl Fentanyl 9822 I Y N-(1-phenethylpiperidin-4-yl)-N-phenylbutyramide, N-(1-phenethylpiperidin-4-yl)-N-phenylbutanamide
Cathinone 1235 I N Constituent of "Khat" plant
Clonitazene 9612 I Y
Codeine methylbromide 9070 I Y
Codeine-N-oxide 9053 I Y
CP-47,497 (5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3- 7297 I N CP-47,497 hydroxycyclohexyl-phenol)
CP-47,497 C8 Homologue (5-(1,1-Dimethyloctyl)-2- 7298 I N CP-47,497 C8 Homologue [(1R,3S)3-hydroxycyclohexyl-phenol)
Cyprenorphine 9054 I Y
Desomorphine 9055 I Y
Dextromoramide 9613 I Y Palfium, Jetrium, Narcolo
Diampromide 9615 I Y
Diethylthiambutene 9616 I Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 3 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Diethyltryptamine 7434 I N DET, N,N-Diethyltryptamine (Positional Isomer: N-Methyl-N-isopropyltryptamine (MiPT))
Difenoxin 9168 I Y Lyspafen
Dihydromorphine 9145 I Y
Dimenoxadol 9617 I Y
Dimepheptanol 9618 I Y
Dimethylthiambutene 9619 I Y
Dimethyltryptamine 7435 I N DMT
Dioxaphetyl butyrate 9621 I Y
Dipipanone 9622 I Y Dipipan, phenylpiperone HCl, Diconal, Wellconal
Drotebanol 9335 I Y Metebanyl, oxymethebanol
Ethylmethylthiambutene 9623 I Y
Etonitazene 9624 I Y
Etorphine (except HCl) 9056 I Y
Etoxeridine 9625 I Y
Fenethylline 1503 I N Captagon,amfetyline,ethyltheophylline amphetamine
Furethidine 9626 I Y
Gamma Hydroxybutyric Acid 2010 I N GHB, gamma hydroxybutyrate, sodium oxybate
Heroin 9200 I Y Diacetylmorphine, diamorphine
Hydromorphinol 9301 I Y
Hydroxypethidine 9627 I Y
Ibogaine 7260 I N Constituent of "Tabernanthe iboga" plant
JWH-018 (also known as AM678) (1-Pentyl-3-(1- 7118 I N JWH-018 and AM-678 naphthoyl)indole)
JWH-019 (1-Hexyl-3-(1-naphthoyl)indole) 7019 I N JWH-019
JWH-073 (1-Butyl-3-(1-naphthoyl)indole) 7173 I N JWH-073
JWH-081 (1-Pentyl-3-(1-(4-methoxynaphthoyl) indole) 7081 I N JWH-081
JWH-122 (1-Pentyl-3-(4-methyl-1-naphthoyl) indole) 7122 I N JWH-122
JWH-200 (1-[2-(4-Morpholinyl)ethyl]-3-(1- 7200 I N JWH-200 naphthoyl)indole)
JWH-203 (1-Pentyl-3-(2-chlorophenylacetyl) indole) 7203 I N JWH-203
JWH-250 (1-Pentyl-3-(2-methoxyphenylacetyl) indole) 6250 I N JWH-250
JWH-398 (1-Pentyl-3-(4-chloro-1-naphthoyl) indole) 7398 I N JWH-398
Ketobemidone 9628 I Y Cliradon
Levomoramide 9629 I Y
Levophenacylmorphan 9631 I Y
Lysergic acid diethylamide 7315 I N LSD, lysergide
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 4 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
MAB-CHMINACA (N-(1-amino-3,3dimethyl-1- 7032 I N MAB-CHMINACA and ADB-CHMINACA oxobutan-2-yl)-1-(cyclohexylmethyl)-1H-indazole-3-carboxamide)
Marihuana 7360 I N Cannabis, marijuana
MDPV (3,4-Methylenedioxypyrovalerone) 7535 I N MDPV
Mecloqualone 2572 I N Nubarene
Mephedrone (4-Methyl-N-methylcathinone) 1248 I N (Positional Isomers: 3-Methyl-methcathinone, Buphedrone, Ethcathinone, N,N-Dimethyl-cathinone)
Mescaline 7381 I N Constituent of "Peyote" cacti
Methaqualone 2565 I N Quaalude, Parest, Somnafac, Opitimil, Mandrax
Methcathinone 1237 I N N-Methylcathinone, "cat"
Methyldesorphine 9302 I Y
Methyldihydromorphine 9304 I Y
Methylone (3,4-Methylenedioxy-N-methylcathinone) 7540 I N Methylone
Morpheridine 9632 I Y
Morphine methylbromide 9305 I Y
Morphine methylsulfonate 9306 I Y
Morphine-N-oxide 9307 I Y
Myrophine 9308 I Y
N,N-Dimethylamphetamine 1480 I N
Naphyrone 1258 I N naphthylpyrovalerone; 1-(naphthalen-2-yl)-2-(pyrrolidin-1-yl)pentan-1-one) (Positional Isomer: α-naphyrone)
N-Benzylpiperazine 7493 I N BZP, 1-benzylpiperazine
N-Ethyl-1-phenylcyclohexylamine 7455 I N PCE
N-Ethyl-3-piperidyl benzilate 7482 I N JB 323
N-Ethylamphetamine 1475 I N NEA
N-Hydroxy-3,4-methylenedioxyamphetamine 7402 I N N-hydroxy MDA
Nicocodeine 9309 I Y
Nicomorphine 9312 I Y Vilan
N-Methyl-3-piperidyl benzilate 7484 I N JB 336
Noracymethadol 9633 I Y
Norlevorphanol 9634 I Y
Normethadone 9635 I Y Phenyldimazone
Normorphine 9313 I Y
Norpipanone 9636 I Y
Para-Fluorofentanyl 9812 I Y China White, fentanyl
Parahexyl 7374 I N Synhexyl,
PB-22 (Quinolin-8-yl 1-pentyl-1H-indole-3-carboxylate) 7222 I N QUPIC; PB-22
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 5 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Pentedrone (α-methylaminovalerophenone) 1246 I N 2-(methylamino)-1-phenylpentan-1-one)(Positional Isomers:3-methylethcathinone (3-MEC), 4-ethylmethcathinone (4-EMC), 4-methylbuphedrone (4-MeMABP;4-MeBP), 3,4-dimethylmethcathinone (3,4-DMMC),N-ethylbuphedrone (NEB),N-ethyl-N-methylcathinone(EMC))
Pentylone 7542 I N bk-MBDP; 1-(1,3-benzodioxol-5-yl)-2-(methylamino)pentan-1-one) (Positional Isomer: dibutylone (bk-DMBDB))
Peyote 7415 I N Cactus which contains mescaline
Phenadoxone 9637 I Y
Phenampromide 9638 I Y
Phenomorphan 9647 I Y
Phenoperidine 9641 I Y Operidine, Lealgin
Pholcodine 9314 I Y Copholco, Adaphol, Codisol, Lantuss, Pholcolin
Piritramide 9642 I Y Piridolan
Proheptazine 9643 I Y
Properidine 9644 I Y
Propiram 9649 I Y Algeril
Psilocybin 7437 I N Constituent of "Magic mushrooms"
Psilocyn 7438 I N Psilocin, constituent of "Magic mushrooms"
Racemoramide 9645 I Y
SR-18 (Also known as RCS-8) (1-Cyclohexylethyl-3-(2- 7008 I N SR-18 and RCS-8 methoxyphenylacetyl) indole)
SR-19 (Also known as RCS-4) (1-Pentyl-3-[(4- 7104 I N SR-19 and RCS-4 methoxy)-benzoyl] indole
Tetrahydrocannabinols 7370 I N THC, Delta-8 THC, Delta-9 THC, dronabinol and others
Thebacon 9315 I Y Acetylhydrocodone, Acedicon, Thebacetyl
Thiofentanyl 9835 I Y Chine white, fentanyl
THJ-2201 [1-(5-fluoropentyl)-1H-indazol-3- 7024 I N THJ-2201 yl](naphthalen-1-yl)methanone
Tilidine 9750 I Y Tilidate, Valoron, Kitadol, Lak, Tilsa
Trimeperidine 9646 I Y Promedolum
UR-144 (1-Pentyl-1H-indol-3-yl)(2,2,3,3- 7144 I N UR-144 tetramethylcyclopropyl)methanone
1-Phenylcyclohexylamine 7460 II N PCP precursor
1-Piperidinocyclohexanecarbonitrile 8603 II N PCC, PCP precursor
4-Anilino-N-phenethyl-4-piperidine (ANPP) 8333 II N ANPP
Alfentanil 9737 II Y Alfenta
Alphaprodine 9010 II Y Nisentil
Amobarbital 2125 II N Amytal, Tuinal
Amphetamine 1100 II N Dexedrine, Adderall, Obetrol
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 6 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Anileridine 9020 II Y Leritine
Bezitramide 9800 II Y Burgodin
Carfentanil 9743 II Y Wildnil
Coca Leaves 9040 II Y
Cocaine 9041 II Y Methyl benzoylecgonine, Crack
Codeine 9050 II Y Morphine methyl ester, methyl morphine
Dextropropoxyphene, bulk (non-dosage forms) 9273 II Y Propoxyphene
Dihydrocodeine 9120 II Y Didrate, Parzone
Dihydroetorphine 9334 II Y DHE
Diphenoxylate 9170 II Y
Ecgonine 9180 II Y Cocaine precursor, in Coca leaves
Ethylmorphine 9190 II Y Dionin
Etorphine HCl 9059 II Y M 99
Fentanyl 9801 II Y Duragesic, Oralet, Actiq, Sublimaze, Innovar
Glutethimide 2550 II N Doriden, Dorimide
Hydrocodone 9193 II Y dihydrocodeinone
Hydromorphone 9150 II Y Dilaudid, dihydromorphinone
Isomethadone 9226 II Y Isoamidone
Levo-alphacetylmethadol 9648 II Y LAAM, long acting methadone, levomethadyl acetate
Levomethorphan 9210 II Y
Levorphanol 9220 II Y Levo-Dromoran
Lisdexamfetamine 1205 II N Vyvanse
Meperidine 9230 II Y Demerol, Mepergan, pethidine
Meperidine intermediate-A 9232 II Y Meperidine precursor
Meperidine intermediate-B 9233 II Y Meperidine precursor, normeperidine
Meperidine intermediate-C 9234 II Y Meperidine precursor
Metazocine 9240 II Y
Methadone 9250 II Y Dolophine, Methadose, Amidone
Methadone intermediate 9254 II Y Methadone precursor
Methamphetamine 1105 II N Desoxyn, D-desoxyephedrine, ICE, Crank, Speed
Methylphenidate 1724 II N Concerta, Ritalin, Methylin
Metopon 9260 II Y
Moramide-intermediate 9802 II Y
Morphine 9300 II Y MS Contin, Roxanol, Oramorph, RMS, MSIR
Nabilone 7379 II N Cesamet
Opium extracts 9610 II Y
Opium fluid extract 9620 II Y
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 7 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Opium poppy 9650 II Y Papaver somniferum
Opium tincture 9630 II Y Laudanum
Opium, granulated 9640 II Y Granulated opium
Opium, powdered 9639 II Y Powdered opium
Opium, raw 9600 II Y Raw opium, gum opium
Oripavine 9330 II Y
Oxycodone 9143 II Y OxyContin, Percocet, Endocet, Roxicodone, Roxicet,
Oxymorphone 9652 II Y Numorphan
Pentobarbital 2270 II N Nembutal
Phenazocine 9715 II Y Narphen, Prinadol
Phencyclidine 7471 II N PCP, Sernylan
Phenmetrazine 1631 II N Preludin
Phenylacetone 8501 II N P2P, phenyl-2-propanone, benzyl methyl ketone
Piminodine 9730 II Y
Poppy Straw 9650 II Y Opium poppy capsules, poppy heads
Poppy Straw Concentrate 9670 II Y Concentrate of Poppy Straw, CPS
Racemethorphan 9732 II Y
Racemorphan 9733 II Y Dromoran
Remifentanil 9739 II Y Ultiva
Secobarbital 2315 II N Seconal, Tuinal
Sufentanil 9740 II Y Sufenta
Tapentadol 9780 II Y
Thebaine 9333 II Y Precursor of many narcotics
Thiafentanil 9729 II Y Thianil
13Beta-ethyl-17beta-hydroxygon-4-en-3-one 4000 III N
17Alpha-methyl-3alpha,17beta-dihydroxy-5alpha- 4000 III N androstane
17Alpha-methyl-3beta,17beta-dihydroxy-5alpha- 4000 III N androstane
17Alpha-methyl-3beta,17beta-dihydroxyandrost-4-ene 4000 III N
17Alpha-methyl-4-hydroxynandrolone (17alpha-methyl- 4000 III N 4-hydroxy-17beta-hydroxyestr-4-en-3-one)
17Alpha-methyl-delta1-dihydrotestosterone (17beta- 4000 III N 17-Alpha-methyl-1-testosterone hydroxy-17alpha-methyl-5alpha-androst-1-en-3-one)
19-Nor-4,9(10)-androstadienedione 4000 III N
19-Nor-4-androstenediol (3beta,17beta-dihydroxyestr-4- 4000 III N ene; 3alpha,17beta-dihydroxyestr-4-ene)
19-Nor-4-androstenedione (estr-4-en-3,17-dione) 4000 III N
19-Nor-5-androstenediol (3beta,17beta-dihydroxyestr-5- 4000 III N ene; 3alpha,17beta-dihydroxyestr-5-ene)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 8 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
19-Nor-5-androstenedione (estr-5-en-3,17-dione) 4000 III N
1-Androstenediol (3beta,17beta-dihydroxy-5alpha- 4000 III N androst-1-ene; 3alpha,17beta-dihydroxy-5alpha-androst-1-ene)
1-Androstenedione (5alpha-androst-1-en-3,17-dione) 4000 III N
3Alpha,17beta-dihydroxy-5alpha-androstane 4000 III N
3Beta,17beta-dihydroxy-5alpha-androstane 4000 III N
4-Androstenediol (3beta,17beta-dihydroxy-androst-4- 4000 III N 4-AD ene)
4-Androstenedione (androst-4-en-3,17-dione) 4000 III N
4-Dihydrotestosterone (17beta-hydroxyandrostan-3- 4000 III N Anabolex, Andractim, Pesomax, Stanolone one)
4-Hydroxy-19-nortestosterone (4,17beta-dihydroxyestr- 4000 III N 4-en-3-one)
4-Hydroxytestosterone (4,17beta-dihydroxyandrost-4- 4000 III N en-3-one)
5-Androstenediol (3beta,17beta-dihydroxy-androst-5- 4000 III N ene)
5-Androstenedione (androst-5-en-3,17-dione) 4000 III N
Amobarbital & noncontrolled active ingred. 2126 III N
Amobarbital suppository dosage form 2126 III N
Anabolic steroids 4000 III N "Body Building" drugs
Androstanedione (5alpha-androstan-3,17-dione) 4000 III N
Aprobarbital 2100 III N Alurate
Barbituric acid derivative 2100 III N Barbiturates not specifically listed
Benzphetamine 1228 III N Didrex, Inapetyl
Bolasterone (7alpha,17alpha-dimethyl-17beta- 4000 III N hydroxyandrost-4-en-3-one)
Boldenone (17beta-hydroxyandrost-1,4-diene-3-one) 4000 III N Equipoise, Parenabol, Vebonol, dehydrotestosterone
Boldione 4000 III N
Buprenorphine 9064 III Y Buprenex, Temgesic, Subutex, Suboxone
Butabarbital (secbutabarbital) 2100 III N Butisol, Butibel
Butalbital 2100 III N Fiorinal, Butalbital with aspirin
Butobarbital (butethal) 2100 III N Soneryl (UK)
Calusterone (7beta,17alpha-dimethyl-17beta- 4000 III N Methosarb hydroxyandrost-4-en-3-one)
Chlorhexadol 2510 III N Mechloral, Mecoral, Medodorm, Chloralodol
Chlorphentermine 1645 III N Pre-Sate, Lucofen, Apsedon, Desopimon
Clortermine 1647 III N Voranil
Clostebol (4-chloro-17beta-hydroxyandrost-4-en-3-one) 4000 III N Alfa-Trofodermin, Clostene, 4-chlorotestosterone
Codeine & isoquinoline alkaloid 90 mg/du 9803 III Y Codeine with papaverine or noscapine
Codeine combination product 90 mg/du 9804 III Y Empirin,Fiorinal,Tylenol,ASA or APAP w/codeine
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 9 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Dehydrochloromethyltestosterone (4-chloro-17beta-hydroxy-17alpha-methylandrost-1,4-dien-3-one)
4000 III N Oral-Turinabol
Delta1-dihydrotestosterone (17beta-hydroxy-5alpha-androst-1-en-3-one)
4000 III N 1-Testosterone
Desoxymethyltestosterone 4000 III N
Dihydrocodeine combination product 90 mg/du 9807 III Y Synalgos-DC, Compal
Dronabinol (synthetic) in sesame oil in soft gelatin capsule as approved by FDA
7369 III N Marinol, synthetic THC in sesame oil/soft gelatin as approved by FDA
Drostanolone (17beta-hydroxy-2alpha-methyl-5alpha-androstan-3-one)
4000 III N Drolban, Masterid, Permastril
Embutramide 2020 III N Tributane
Ethylestrenol (17alpha-ethyl-17beta-hydroxyestr-4-ene) 4000 III N Maxibolin, Orabolin, Durabolin-O, Duraboral
Ethylmorphine combination product 15 mg/du 9808 III Y
Fluoxymesterone (9-fluoro-17alpha-methyl-11beta,17beta-dihydroxyandrost-4-en-3-one)
4000 III N Anadroid-F, Halotestin, Ora-Testryl
Formebolone (2-formyl-17alpha-methyl-11alpha,17beta-dihydroxyandrost-1,4-dien-3-one)
4000 III N Esiclene, Hubernol
Furazabol (17alpha-methyl-17beta-hydroxyandrostano[2,3-c]-furazan)
4000 III N Frazalon, Miotolon, Qu Zhi Shu
Gamma Hydroxybutyric Acid preparations 2012 III N Xyrem
Ketamine 7285 III N Ketaset, Ketalar, Special K, K
Lysergic acid 7300 III N LSD precursor
Lysergic acid amide 7310 III N LSD precursor
Mestanolone (17alpha-methyl-17beta-hydroxy-5alpha-androstan-3-one)
4000 III N Assimil, Ermalone, Methybol, Tantarone
Mesterolone (1alpha-methyl-17beta-hydroxy-5alpha-androstan-3-one)
4000 III N Androviron, Proviron, Testiwop
Methandienone (17alpha-methyl-17beta-hydroxyandrost-1,4-diene-3-one)
4000 III N Dianabol, Metabolina, Nerobol, Perbolin
Methandriol (17alpha-methyl-3beta,17beta-dihydroxyandrost-5-ene)
4000 III N Sinesex, Stenediol, Troformone
Methasterone (2alpha,17alpha-dimethyl-5alpha-androstan-17beta-ol-3-one)
4000 III N Methasterone
Methenolone (1-methyl-17beta-hydroxy-5alpha-androst-1-en-3-one)
4000 III N Primobolan, Primobolan Depot, Primobolan S
Methyldienolone (17alpha-methyl-17beta-hydroxyestr-4,9(10)-dien-3-one)
4000 III N
Methyltestosterone (17alpha-methyl-17beta-hydroxyandrost-4-en-3-one)
4000 III N Android, Oreton, Testred, Virilon
Methyltrienolone (17alpha-methyl-17beta-hydroxyestr-4,9,11-trien-3-one)
4000 III N Metribolone
Methyprylon 2575 III N Noludar
Mibolerone (7alpha,17alpha-dimethyl-17beta-hydroxyestr-4-en-3-one)
4000 III N Cheque, Matenon
Morphine combination product/50 mg/(100 ml or 100 gm)
9810 III Y
Nalorphine 9400 III Y Nalline
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 10 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Nandrolone (17beta-hydroxyestr-4-en-3-one) 4000 III N Deca-Durabolin, Durabolin, Durabolin-50
Norbolethone (13beta,17alpha-diethyl-17beta- 4000 III N Genabol hydroxygon-4-en-3-one)
Norclostebol (4-chloro-17beta-hydroxyestr-4-en-3-one 4000 III N Anabol-4-19, Lentabol
Norethandrolone (17alpha-ethyl-17beta-hydroxyestr-4- 4000 III N Nilevar, Pronabol, Solevar en-3-one)
Normethandrolone (17alpha-methyl-17beta- 4000 III N Lutenin, Matronal, Orgasteron hydroxyestr-4-en-3-one)
Opium combination product 25 mg/du 9809 III Y Paregoric, other combination products
Oxandrolone (17alpha-methyl-17beta-hydroxy-2-oxa- 4000 III N Anavar, Lonavar, Oxandrin, Provitar, Vasorome 5alpha-androstan-3-one)
Oxymesterone (17alpha-methyl-4,17beta- 4000 III N Anamidol, Balnimax, Oranabol, Oranabol 10 dihydroxyandrost-4-en-3-one)
Oxymetholone (17alpha-methyl-2-hydroxymethylene- 4000 III N Anadrol-50, Adroyd, Anapolon, Anasteron, Pardroyd 17beta-hydroxy-5alpha-androstan-3-one)
Pentobarbital & noncontrolled active ingred. 2271 III N FP-3
Pentobarbital suppository dosage form 2271 III N WANS
Perampanel 2261 III N Fycompa, [2-(2-oxo-l-phenyl-5-pyridin-2-yl-l ,2-dihydropyridin-3-yl) benzonitrile ]
Phendimetrazine 1615 III N Plegine, Prelu-2, Bontril, Melfiat, Statobex
Prostanozol (17beta-hydroxy-5alpha-androstano[3,2- 4000 III N Prostanozol c]pyrazole)
Secobarbital & noncontrolled active ingred 2316 III N
Secobarbital suppository dosage form 2316 III N
Stanozolol (17alpha-methyl-17beta-hydroxy-5alpha- 4000 III N Winstrol, Winstrol-V androst-2-eno[3,2-c]-pyrazole)
Stenbolone (17beta-hydroxy-2-methyl--5alpha-androst- 4000 III N 1-en-3-one)
Stimulant compounds previously excepted 1405 III N Mediatric
Sulfondiethylmethane 2600 III N
Sulfonethylmethane 2605 III N
Sulfonmethane 2610 III N
Talbutal 2100 III N Lotusate
Testolactone (13-hydroxy-3-oxo-13,17-secoandrosta- 4000 III N Teolit, Teslac 1,4-dien-17-oic acid lactone)
Testosterone (17beta-hydroxyandrost-4-en-3-one) 4000 III N Android-T, Androlan, Depotest, Delatestryl
Tetrahydrogestrinone (13beta,17alpha-diethyl-17beta- 4000 III N THG hydroxygon-4,9,11-trien-3-one)
Thiamylal 2100 III N Surital
Thiopental 2100 III N Pentothal
Tiletamine & Zolazepam Combination Product 7295 III N Telazol
Trenbolone (17beta-hydroxyestr-4,9,11-trien-3-one) 4000 III N Finaplix-S, Finajet, Parabolan
Vinbarbital 2100 III N Delvinal, vinbarbitone
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 11 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Alfaxalone 2731 IV N Alfaxan, 5α-pregnan-3α-ol-11,20-dione
Alprazolam 2882 IV N Xanax
Barbital 2145 IV N Veronal, Plexonal, barbitone
Bromazepam 2748 IV N Lexotan, Lexatin, Lexotanil
Butorphanol 9720 IV N Stadol, Stadol NS, Torbugesic, Torbutrol
Camazepam 2749 IV N Albego, Limpidon, Paxor
Carisoprodol 8192 IV N Soma
Cathine 1230 IV N Constituent of "Khat" plant, (+)-norpseudoephedrine
Chloral betaine 2460 IV N Beta Chlor
Chloral hydrate 2465 IV N Noctec
Chlordiazepoxide 2744 IV N Librium, Libritabs, Limbitrol, SK-Lygen
Clobazam 2751 IV N Urbadan, Urbanyl
Clonazepam 2737 IV N Klonopin, Clonopin
Clorazepate 2768 IV N Tranxene
Clotiazepam 2752 IV N Trecalmo, Rize, Clozan, Veratran
Cloxazolam 2753 IV N Akton, Lubalix, Olcadil, Sepazon
Delorazepam 2754 IV N
Dexfenfluramine 1670 IV N Redux
Dextropropoxyphene dosage forms 9278 IV Y Darvon, propoxyphene, Darvocet, Propacet
Diazepam 2765 IV N Valium, Diastat
Dichloralphenazone 2467 IV N Midrin, dichloralantipyrine
Diethylpropion 1610 IV N Tenuate, Tepanil
Difenoxin 1 mg/25 ug AtSO4/du 9167 IV Y Motofen
Eluxadoline 9725 IV N VIBERZI
Estazolam 2756 IV N ProSom, Domnamid, Eurodin, Nuctalon
Ethchlorvynol 2540 IV N Placidyl
Ethinamate 2545 IV N Valmid, Valamin
Ethyl loflazepate 2758 IV N
Fencamfamin 1760 IV N Reactivan
Fenfluramine 1670 IV N Pondimin, Ponderal
Fenproporex 1575 IV N Gacilin, Solvolip
Fludiazepam 2759 IV N
Flunitrazepam 2763 IV N Rohypnol, Narcozep, Darkene, Roipnol
Flurazepam 2767 IV N Dalmane
Fospropofol 2138 IV N Lusedra
Halazepam 2762 IV N Paxipam
Haloxazolam 2771 IV N
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 12 of 14
DEA CSA
SUBSTANCE NUMBER SCH NARC OTHER NAMES
Ketazolam 2772 IV N Anxon, Loftran, Solatran, Contamex
Loprazolam 2773 IV N
Lorazepam 2885 IV N Ativan
Lorcaserin 1625 IV N Belviq
Lormetazepam 2774 IV N Noctamid
Mazindol 1605 IV N Sanorex, Mazanor
Mebutamate 2800 IV N Capla
Medazepam 2836 IV N Nobrium
Mefenorex 1580 IV N Anorexic, Amexate, Doracil, Pondinil
Meprobamate 2820 IV N Miltown, Equanil, Micrainin, Equagesic, Meprospan
Methohexital 2264 IV N Brevital
Methylphenobarbital (mephobarbital) 2250 IV N Mebaral, mephobarbital
Midazolam 2884 IV N Versed
Modafinil 1680 IV N Provigil
Nimetazepam 2837 IV N Erimin
Nitrazepam 2834 IV N Mogadon
Nordiazepam 2838 IV N Nordazepam, Demadar, Madar
Oxazepam 2835 IV N Serax, Serenid-D
Oxazolam 2839 IV N Serenal, Convertal
Paraldehyde 2585 IV N Paral
Pemoline 1530 IV N Cylert
Pentazocine 9709 IV N Talwin, Talwin NX, Talacen, Talwin Compound
Petrichloral 2591 IV N Pentaerythritol chloral, Periclor
Phenobarbital 2285 IV N Luminal, Bellergal-S
Phentermine 1640 IV N Ionamin, Fastin, Adipex-P, Obe-Nix, Zantryl
Pinazepam 2883 IV N Domar
Pipradrol 1750 IV N Detaril, Stimolag Fortis
Prazepam 2764 IV N Centrax
Quazepam 2881 IV N Doral
Sibutramine 1675 IV N Meridia
SPA 1635 IV N 1-dimethylamino-1,2-diphenylethane, Lefetamine
Suvorexant 2223 IV N MK-4305, [(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone
Temazepam 2925 IV N Restoril
Tetrazepam 2886 IV N Myolastan, Musaril
Tramadol (2-[(dimethylamino)methyl]-1-(3- 9752 IV Y Tramadol methoxyphenyl)cyclohexanol)
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 13 of 14
SUBSTANCE
DEA
NUMBER
CSA
SCH NARC OTHER NAMES
Triazolam 2887 IV N Halcion
Zaleplon 2781 IV N Sonata
Zolpidem 2783 IV N Ambien, Ivadal, Stilnoct, Stilnox
Zopiclone 2784 IV N Lunesta
Brivaracetam 2710 V N BRV, UCB-34714, Briviact, ((2S)-2-[(4R)-2-oxo-4-propylpyrrolidin-1-yl] butanamide)
Codeine preparations - 200 mg/(100 ml or 100 gm) V Y Cosanyl,Robitussin A-C,Cheracol,Cerose,Pediacof
Difenoxin preparations - 0.5 mg/25 ug AtSO4/du V Y Motofen
Dihydrocodeine preparations 100mg/(100 ml or 100 V Y Cophene-S, various others gm)
Diphenoxylate preparations 2.5 mg/25 ug AtSO4 V Y Lomotil, Logen
Ethylmorphine preparations 100 mg/(100 ml or 100 gm) V Y
Ezogabine 2779 V N Potiga
Lacosamide 2746 V N Vimpat
Opium preparations - 100 mg/(100 ml or 100 gm) V Y Parepectolin, Kapectolin PG, Kaolin Pectin P.G.
Pregabalin 2782 V N Lyrica
Pyrovalerone 1485 V N Centroton, Thymergix
Abbreviations: "NARC"= Narcotic, "CSA SCH"= CSA Schedule
Controlled Substances - by CSA Schedule
29-Aug-16 Page 14 of 14
List I and List II Regulated C
hemicals
1. Alphabetical Order 2. DEA Number 3. List Number 4. Illicit Uses and Threshold Quantities
List I and II Regulated Chemicals
- Alphabetical Order -
LIST DEA EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
ACETIC ANHYDRIDE II 8519 Pub. L. 100-690
3/18/1989
ACETONE II 6532 Pub. L. 100-690
3/18/1989
N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690
3/18/1989
ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690
3/18/1989
BENZALDEHYDE I 8256 Pub. L. 103-200
4/17/1994
BENZYL CHLORIDE II 8570 Pub. L. 100-690
3/18/1989
BENZYL CYANIDE I 8735 Pub. L. 100-690
3/18/1989
gamma-BUTYROLACTONE I 2011 Pub. L. 106-172
2/18/2000
EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690
3/18/1989
EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200
4/17/1994
EPHEDRINE-remove exemption for OTC combination products and establish a 24 g retail threshold. Threshold remains zero for single entity products. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, 1313
I 8113 Pub. L. 104-237
10/3/1996
ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690
3/18/1989
ERGOCRISTINE I 8612 76 FR 17778 5/2/2011
ERGOTAMINE & salts I 8676 Pub. L. 100-690
3/18/1989
ETHYLAMINE & salts I 8678 Pub. L. 101-647
2/27/1991
N-ETHYLEPHEDRINE - superseded by 1994 action I Pub. L. 101-647
2/27/1991
N-ETHYLEPHEDRINE REMOVED Pub. L. 103-200
4/17/1994
ETHYL ETHER II 6584 Pub. L. 100-690
3/18/1989
N-ETHYLPSEUDOEPHEDRINE - superseded by 1994 action I Pub. L. 101-647
2/27/1991
N-ETHYLPSEUDOEPHEDRINE REMOVED Pub. L. 103-200
4/17/1994
HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992
HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237
10/3/1996
* Remain in Schedule III
List I and II Regulated Chemicals - Alphabetical Order
29-Aug-16 Page 1 of 3
REGULATED CHEMICAL
LIST
NUMBER
DEA
NUMBER CITATION
EFFECTIVE
DATE
HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690
3/18/1989
HYDRIODIC ACID I 6695 Pub. L. 101-647
2/27/1991
HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, calcium hypophosphite, iron hypophosphite, potassium hypophosphite, manganese hypophosphite, magnesium hypophosphite, and sodium hypophosphite)
I 6797 66 FR 52670 11/16/2001
IODINE - superseded by 2007 action II 6699 Pub. L. 104-237
10/3/1996
IODINE I 6699 72 FR 35920 8/1/2007
ISOSAFROLE I 8704 Pub. L. 101-647
2/27/1991
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers-superseded
I 7300 Pub. L. 101-647
2/27/1991
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers* REMOVED 7300 Pub. L. 103-200
4/17/1994
METHYLAMINE and salts I 8520 Pub. L. 101-647
2/27/1991
3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690
3/18/1989
N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647
2/27/1991
METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690
3/18/1989
METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995
N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical isomers
I 8119 Pub. L. 101-647
2/27/1991
NITROETHANE I 6724 Pub. L. 103-200
4/17/1994
NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690
3/18/1989
N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007
PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690
3/18/1989
PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690
3/18/1989
PHENYLPROPANOLAMINE-remove exemption for certain OTC transactions. Retail threshold of 24 g established for products not distributed in blister packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
I 1225 Pub. L. 104-237
10/3/1997
PIPERIDINE and salts I 2704 Pub. L. 100-690
3/18/1989
PIPERONAL I 8750 Pub. L. 101-647
2/27/1991
POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690
3/18/1989
PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647
2/27/1991
* Remain in Schedule III
List I and II Regulated Chemicals - Alphabetical Order
29-Aug-16 Page 2 of 3
LIST DEA EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100- 3/18/1989 690
PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. I 8112 Pub. L. 104- 10/3/1997 Retail threshold of 24 g established for products not distributed in blister 237 packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001
SAFROLE (includes sassafras oil) I 8323 Pub. L. 101- 2/27/1991 647
SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006
SULFURIC ACID II 6552 57 FR 43614 10/22/1992
TOLUENE II 6594 Pub. L. 100- 3/18/1989 690
WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001
* Remain in Schedule III
List I and II Regulated Chemicals - Alphabetical Order
Page 3 of 3 29-Aug-16
List I and II Regulated Chemicals
- by DEA Number -
LIST DEA EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
N-ETHYLEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991
N-ETHYLEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
N-ETHYLPSEUDOEPHEDRINE - superseded by 1994 action I Pub. L. 101-647 2/27/1991
N-ETHYLPSEUDOEPHEDRINE REMOVED Pub. L. 103-200 4/17/1994
PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE-remove exemption for certain OTC transactions. I 1225 Pub. L. 104-237 10/3/1997 Retail threshold of 24 g established for products not distributed in blister packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
gamma-BUTYROLACTONE I 2011 Pub. L. 106-172 2/18/2000
PIPERIDINE and salts I 2704 Pub. L. 100-690 3/18/1989
ACETONE II 6532 Pub. L. 100-690 3/18/1989
HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992
HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237 10/3/1996
SULFURIC ACID II 6552 57 FR 43614 10/22/1992
POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690 3/18/1989
ETHYL ETHER II 6584 Pub. L. 100-690 3/18/1989
SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006
TOLUENE II 6594 Pub. L. 100-690 3/18/1989
HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690 3/18/1989
HYDRIODIC ACID I 6695 Pub. L. 101-647 2/27/1991
IODINE - superseded by 2007 action II 6699 Pub. L. 104-237 10/3/1996
IODINE I 6699 72 FR 35920 8/1/2007
METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690 3/18/1989
METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995
NITROETHANE I 6724 Pub. L. 103-200 4/17/1994
RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001
WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001
HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, I 6797 66 FR 52670 11/16/2001 calcium hypophosphite, iron hypophosphite, potassium hypophosphite, manganese hypophosphite, magnesium hypophosphite, and sodium hypophosphite)
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers- I 7300 Pub. L. 101-647 2/27/1991 superseded
D-LYSERGIC ACID, salts, optical isomers, & salts of optical isomers* REMOVED 7300 Pub. L. 103-200 4/17/1994
PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100-690 3/18/1989
* Remain in Schedule III
List I and II Regulated Chemicals - by DEA Number
Page 1 of 2 29-Aug-16
REGULATED CHEMICAL
LIST
NUMBER
DEA
NUMBER CITATION
EFFECTIVE
DATE
PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. Retail threshold of 24 g established for products not distributed in blister packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
I 8112 Pub. L. 104-237 10/3/1997
EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690 3/18/1989
EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200 4/17/1994
EPHEDRINE-remove exemption for OTC combination products and establish I 8113 Pub. L. 104-237 10/3/1996 a 24 g retail threshold. Threshold remains zero for single entity products. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, 1313
N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647 2/27/1991
N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical I 8119 Pub. L. 101-647 2/27/1991 isomers
BENZALDEHYDE I 8256 Pub. L. 103-200 4/17/1994
NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690 3/18/1989
SAFROLE (includes sassafras oil) I 8323 Pub. L. 101-647 2/27/1991
PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647 2/27/1991
N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007
3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690 3/18/1989
ACETIC ANHYDRIDE II 8519 Pub. L. 100-690 3/18/1989
METHYLAMINE and salts I 8520 Pub. L. 101-647 2/27/1991
N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690 3/18/1989
ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690 3/18/1989
BENZYL CHLORIDE II 8570 Pub. L. 100-690 3/18/1989
ERGOCRISTINE I 8612 76 FR 17778 5/2/2011
ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690 3/18/1989
ERGOTAMINE & salts I 8676 Pub. L. 100-690 3/18/1989
ETHYLAMINE & salts I 8678 Pub. L. 101-647 2/27/1991
ISOSAFROLE I 8704 Pub. L. 101-647 2/27/1991
BENZYL CYANIDE I 8735 Pub. L. 100-690 3/18/1989
PIPERONAL I 8750 Pub. L. 101-647 2/27/1991
PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690 3/18/1989
* Remain in Schedule III
List I and II Regulated Chemicals - by DEA Number
Page 2 of 2 29-Aug-16
List I and II Regulated Chemicals
- by List Number -
LIST DEA EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
N-ACETYLANTHRANILIC ACID, salts & esters I 8522 Pub. L. 100-690 3/18/1989
ANTHRANILIC ACID, salts & esters I 8530 Pub. L. 100-690 3/18/1989
BENZALDEHYDE I 8256 Pub. L. 103-200 4/17/1994
BENZYL CYANIDE I 8735 Pub. L. 100-690 3/18/1989
gamma-BUTYROLACTONE I 2011 Pub. L. 106-172 2/18/2000
EPHEDRINE, salts, optical isomers, & salts of optical isomers I 8113 Pub. L. 100-690 3/18/1989
EPHEDRINE - remove exemption for OTC single entity drug product I 8113 Pub. L. 103-200 4/17/1994
EPHEDRINE remove exemption for OTC ephedrine combination products I 8113 Pub. L. 104-237 10/3/1996 and establish a 24 g retail threshold. Threshold remains zero for single entity products. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, 1313.
ERGONOVINE or ERGOMETRINE & salts I 8675 Pub. L. 100-690 3/18/1989
ERGOCRISTINE and its salts I 8612 76 FR 17778 5/2/2011
ERGOTAMINE & salts I 8676 Pub. L. 100-690 3/18/1989
ETHYLAMINE & salts I 8678 Pub. L. 101-647 2/27/1991
HYDRIODIC ACID I 6695 Pub. L. 101-647 2/27/1991
HYPOPHOSPHOROUS ACID, salts (Including ammonium hypophosphite, I 6797 66 FR 52670 11/16/2001 calcium hypophosphite, iron hypophosphite, potassium hypophosphite, manganese hypophosphite, magnesium hypophosphite, and sodium hypophosphite)
IODINE I 6699 72 FR 35920 8/1/2007
ISOSAFROLE I 8704 Pub. L. 101-647 2/27/1991
METHYLAMINE and salts I 8520 Pub. L. 101-647 2/27/1991
3,4-METHYLENEDIOXYPHENYL-2-PROPANONE I 8502 Pub. L. 100-690 3/18/1989
N-METHYLEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8115 Pub. L. 101-647 2/27/1991
N-METHYLPSEUDOEPHEDRINE, salts, optical isomers, salts of optical I 8119 Pub. L. 101-647 2/27/1991 isomers
NITROETHANE I 6724 Pub. L. 103-200 4/17/1994
NORPSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8317 Pub. L. 100-690 3/18/1989
N-PHENETHYL-4-PIPERIDONE (NPP) I 8332 73 FR 43355 4/23/2007
PHENYLACETIC ACID, esters, and salts I 8791 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE, salts, optical isomers, & salts of optical isomers I 1225 Pub. L. 100-690 3/18/1989
PHENYLPROPANOLAMINE -remove exemption for certain OTC I 1225 Pub. L. 104-237 10/3/1997 transactions. Retail threshold of 24 g established for products not distributed in blister packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
List I and II Regulated Chemicals - by List Number
29-Aug-16 Page 1 of 2
LIST DEA EFFECTIVE
REGULATED CHEMICAL NUMBER NUMBER CITATION DATE
PIPERIDINE and salts I 2704 Pub. L. 100-690 3/18/1989
PIPERONAL I 8750 Pub. L. 101-647 2/27/1991
PROPIONIC ANHYDRIDE I 8328 Pub. L. 101-647 2/27/1991
PSEUDOEPHEDRINE, salts, optical isomers, & salts of optical isomers I 8112 Pub. L. 100-690 3/18/1989
PSEUDOEPHEDRINE -remove exemption for certain OTC transactions. I 8112 Pub. L. 104-237 10/3/1997 Retail threshold of 24 g established for products not distributed in blister packs. Mail order report requirements imposed. For more info, see 21 CFR Parts 1309, 1310, and 1313.
RED PHOSPHORUS I 6795 66 FR 52670 11/16/2001
SAFROLE (includes sassafras oil) I 8323 Pub. L. 101-647 2/27/1991
WHITE PHOSPHORUS (Other names: YELLOW PHOSPHORUS) I 6796 66 FR 52670 11/16/2001
ACETIC ANHYDRIDE II 8519 Pub. L. 100-690 3/18/1989
ACETONE II 6532 Pub. L. 100-690 3/18/1989
BENZYL CHLORIDE II 8570 Pub. L. 100-690 3/18/1989
ETHYL ETHER II 6584 Pub. L. 100-690 3/18/1989
HYDROCHLORIC ACID (including anhydrous hydrogen chloride) II 6545 57 FR 43614 10/22/1992
HYDROCHLORIC GAS (anhydrous hydrogen chloride) II 6545 Pub. L. 104-237 10/3/1996
HYDRIODIC ACID - superseded by 1990 action II 6695 Pub. L. 100-690 3/18/1989
IODINE - superseded by 2007 action II 6699 Pub. L. 104-237 10/3/1996
METHYL ETHYL KETONE (MEK) or 2-BUTANONE II 6714 Pub. L. 100-690 3/18/1989
METHYL ISOBUTYL KETONE (MIBK) II 6715 60 FR 19509 5/19/1995
POTASSIUM PERMANGANATE II 6579 Pub. L. 100-690 3/18/1989
SODIUM PERMANGANATE II 6588 71 FR 60823 12/18/2006
SULFURIC ACID II 6552 57 FR 43614 10/22/1992
TOLUENE II 6594 Pub. L. 100-690 3/18/1989
List I and II Regulated Chemicals - by List Number
29-Aug-16 Page 2 of 2
=
=
DOM
ESTI
C
IMPO
RTS
&EX
PORT
S
KILOGRAMS
1 and its salts 2 and its salts and esters 3 and its salts, optical isomers, and salts of optical isomers 4 Exports only, to all Western Hemisphere except Canada 5 Exports to all South American countries & Panama - Domestic for HCI gas 6 Threshold for HCI acid and sulfuric acid is 50 gallons, the equivalent weight in kilograms is shown 7 For pseudoephedrine, phenylpropanolamine and ephedrine drug products, see 21 USC § 802(45)(A) and 21 C.F.R. Part 1314 N/C = Not Controlled
Amph
etam
ine
Coca
ine
N,N
-Dim
ethy
lam
phet
amin
e
Ethy
lam
phet
amin
e
Fent
anyl
& a
nalo
gues
GHB
Hero
in
LSD
MDA
MDE
MDM
A
Met
ham
phet
amin
e
Met
haqu
alon
e
Met
hcat
hino
ne
4-M
ethy
lam
inor
ex
Phen
cycl
idin
e (P
CP)
Phen
yl-2
-pro
pano
ne
1. N-Acetylanthranilic acid 2 40 40
2. Anthranilic acid 2 30 30
3. Benzaldehyde 4 4
4. Benzyl cyanide 1 1
5. Ephedrine 3&7 0 0
6. Ergocristine 1 0 0
7. Ergonovine 1 0.010 0.010
8. Ergotamine 1 0.020 0.020
9. Ethylamine 1 1 1
10. gamma-Butyrolactone (GBL) 0 0
11. Hydriodic acid 1.7 1.7
12. Hypophosphorous acid 1 0 0
13. Iodine 0 0
14. Isosafrole 4 4
15. Methylamine 1 1 1
16. 3,4-Methylenedioxyphenyl-2-propanone 4 4
17. N-Methylephedrine 3 1 1
18. N-Methylpseudoephedrine 3 1 1
19. N-phenethyl-4-piperidone (NPP) 0 0
20. Nitroethane 2.5 2.5
21. Norpseudoephedrine 3 2.5 2.5
22. Phenylacetic acid 2 1 1
23. Phenylpropanolamine 3&7 0 0
24. Phosphorus (red) 0 0
25. Phosphorus (white or yellow) 0 0
26. Piperidine 1 0.500 0.500
27. Piperonal (heliotropin) 4 4
28. Propionic anhydride 0.001 0.001
29. Pseudoephedrine 3&7 0 0 30. Safrole 4 4
31. Acetic anhydride 1,023 1,023
32. Acetone 150 1,500
33. Benzyl chloride 1 4
34. Ethyl ether 135.8 1,364
35. Hydrochloric acid 5&6 N/C 222.3
35a. Hydrogen chloride gas 5&6 0 27
36. Methyl ethyl ketone (2-Butanone) 145 1,455
37. Methyl isobutyl ketone 4 N/C 1,523
38. Potassium permanganate 55 500
39. Sodium permanganate 55 500
40. Sulfuric acid 5&6 N/C 347
41. Toluene 159 1,591
LIST
ILI
ST II
CONTROLLED SUBSTANCE PRODUCED
THRE
SHO
LDS
Listed Chemicals Regulated Under the Controlled Substances Act
See 21 C.F.R. §§ 1309, 1310, 1313 and 1314 for details
January 2016 Reagent
Precursor = Solvent