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human Q standard turnaround time ● agonist radioligand
FAMILY ASSAY FORMAT ITEM # GPCR ADENOSINE A2A ● 0004 ADRENERGIC alpha1A 2338
alpha2A 0013beta1 ● 0018beta2 ● 0020
CANNABINOID CB1 ● 0036CB2 ● 0037
CHOLECYSTOKININ CCK1 (CCKA) ● 0039 DOPAMINE D1 0044
D2S ● 1322 ENDOTHELIN ETA ● 0054 HISTAMINE H1 0870
H2 1208 MUSCARINIC M1 0091
M2 0093M3 0095
OPIOID & OPIOID-LIKE delta2 (DOP) ● 0114kappa (KOP) ● 1971mu (MOP) ● 0118
SEROTONIN 5-HT1A ● 01315-HT1B 01325-HT2A ● 04715-HT2B ● 1333
VASOPRESSIN V1a ● 0159
TRANSPORTERS DOPAMINE dopamine
transporter0052
FAMILY ASSAY FORMAT ITEM # NOREPINEPHRINE norepinephrine
transporter0355
SEROTONIN 5-HT transporter 0439
ION CHANNELS GABA CHANNELS BZD (central) ● 0028 GLUTAMATE CHANNELS NMDA 0066 NICOTINIC CHANNELS N neuronal α4β2 ● 3029 SEROTONIN CHANNELS 5-HT3 0411 Ca2+ CHANNELS Ca2+ channel
(L, dihydropyridine site)0161
K+ CHANNELS hERG (membrane preparation)
1868
KV channel 0166 Na+ CHANNELS Na+ channel (site 2) 0169
NUCLEAR RECEPTORS STEROID NUCLEAR RECEPTORS
AR ● 0933GR ● 0469
KINASES CTK Lck kinase 2906
OTHER NON-KINASE ENZYMES AA METABOLISM COX1 0726
COX2 0727 MONOAMINE & NEUROTRANSMITTER
acetylcholinesterase 0363MAO-A 0443
PHOSPHODIESTERASES PDE3A 2432PDE4D2 2434
SafetyScreen44™ PanelAs a leader in safety pharmacology, Eurofins Pharma Discovery Services offers the SafetyScreen44™ panel to enable early identification of significant off-target interactions with your compound. All 44 selected targets, recommended by 4 major pharmaceutical companies (Bowes et al. 2012), are gathered in a cost-effective panel that brings together both robustness (each assay is HTS-compatible) and the strategic choice of information-rich targets.
Ref. P270
Suggested testing: 10 µM (n=2)
Q 10 business days
PharmaDiscovery Services
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