infrequently used combination antiretrovirals · colorado aids education and training center...

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Colorado AIDS Education and Training Center University of Colorado • Anschutz Medical Campus 12631 E. 17th Avenue • MS A089 • Aurora, CO 80045 TEL: 303-724-0646 • FAX: 303-724-7297 • www.caetc.org Developed by Lisa Lawrence, MSW; and Steven Johnson, MD HIV Medication Guide for Quick Reference Reviewers: Jasjit Gill, PharmD, University of Colorado Hospital ID Pharmacy Jacob Langness, PharmD, University of Colorado Hospital ID Pharmacy Judith Bagley, RPh, Denver Health Medical Center ID Pharmacy Combination Antiretrovirals Complera (FTC+RPV+TDF) Combivir(3TC+AZT) Atripla (EFV+FTC+TDF) FDA Pregnancy Category D Stribild (EVG+COBI+FTC+TDF) Epzicom (ABC+3TC) Trizivir (ABC+3TC+AZT) Truvada (FTC+TDF) Triumeq (ABC+DTG+3TC) Aptivus* (tipranavir, TPV) Crixivan (indinavir, IDV) Invirase (saquinavir hard gel capsules, SQV) Videx EC*(didanosine, ddl) Rescriptor (delavirdine, DLV) Zerit*(stavudine, d4T) Protease Inhibitors (PI) Infrequently Used Evotaz (ATV+COBI) Prezcobix (DRV+COBI) Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTI) Descovy (FTC+TAF) Odefsey (FTC+RPV+TAF) Genvoya (EVG+COBI+FTC+TAF) Nucleoside/Nucleotide Analogue Reverse Transcriptase Inhibitors (NRTI) Vitekta* (elvitegravir, EVG) Integrase Inhibitors

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Page 1: Infrequently Used Combination Antiretrovirals · Colorado AIDS Education and Training Center University of Colorado • Anschutz Medical Campus 12631 E. 17th Avenue • MS A089 •

Colorado AIDS Education and Training Center

University of Colorado • Anschutz Medical Campus 12631 E. 17th Avenue • MS A089 • Aurora, CO 80045

TEL: 303-724-0646 • FAX: 303-724-7297 • www.caetc.org Developed by Lisa Lawrence, MSW; and Steven Johnson, MD

HIV Medication Guide for

Quick Reference

Reviewers: Jasjit Gill, PharmD, University of Colorado Hospital ID PharmacyJacob Langness, PharmD, University of Colorado Hospital ID Pharmacy

Judith Bagley, RPh, Denver Health Medical Center ID Pharmacy

Combination AntiretroviralsComplera

(FTC+RPV+TDF)Combivir†

(3TC+AZT)Atripla

(EFV+FTC+TDF)

FDA Pregnancy Category D

Stribild(EVG+COBI+FTC+TDF)

Epzicom▲

(ABC+3TC)

Trizivir †(ABC+3TC+AZT)

Truvada(FTC+TDF)

Triumeq(ABC+DTG+3TC)

Aptivus*(tipranavir, TPV)

Crixivan(indinavir, IDV)

Invirase(saquinavir hard gel

capsules, SQV)

Videx EC*†(didanosine, ddl)

Rescriptor(delavirdine, DLV)

Zerit*†(stavudine, d4T)

Protease Inhibitors (PI)

Infrequently Used

Evotaz(ATV+COBI)

Prezcobix(DRV+COBI)

Non-Nucleoside ReverseTranscriptase Inhibitors (NNRTI)

Descovy(FTC+TAF)

Odefsey(FTC+RPV+TAF)

Genvoya(EVG+COBI+FTC+TAF)Nucleoside/Nucleotide Analogue Reverse Transcriptase Inhibitors (NRTI)

Vitekta*(elvitegravir, EVG)

Integrase Inhibitors

Page 2: Infrequently Used Combination Antiretrovirals · Colorado AIDS Education and Training Center University of Colorado • Anschutz Medical Campus 12631 E. 17th Avenue • MS A089 •

Intelence (etravirine, ETV)

Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTI)

Sustiva(efavirenz, EFV)

FDA Pregnancy Category D

All pills shown in actual size. Medication brand names appear in bold. Generic names and commonly used abbreviations appear in parentheses.Bioavailability and indications between formulations may be different.

Integrase Inhibitors

Boosting Agents

Viramune*†(nevirapine, NVP)

Edurant(rilpivirine, RPV)

Retrovir*†(zidovudine, AZT, ZDV)

Nucleoside/Nucleotide Analogue Reverse Transcriptase Inhibitors (NRTI)

Emtriva*(emtricitabine, FTC)

Epivir*†(lamivudine, 3TC)

Viread* (tenofovir, TDF)

Ziagen*†(abacavir, ABC)

Norvir*(ritonavir, RTV)

05/16

Protease Inhibitors (PI)

Kaletra*(lopinavir/ritonavir, LPV/r)

Viracept*(nelfinavir, NFV)

Lexiva*(fosamprenavir, FPV)

Reyataz*(atazanavir, ATV)

Prezista*(darunavir, DRV)

Isentress▲*(raltegravir, RAL)

Tivicay(dolutegravir, DTG)

Tybost(cobicistat, COBI)

*Also available in liquid or powder form. † Generic formulation available. ▲Chewable form available.

Entry InhibitorsFuzeon

(enfuvirtide, T-20)Fusion Inhibitor

Selzentry(maraviroc, MVC) CCR5 Antagonist