Transcript

Diapositive 1

One-pot total synthesis of K1 HGF domain

85 Aa3 disulfide bridgesK1K2K3K4Na chainSS

K1 weak MET Tyrosine kinase receptor agonist (Holmes, O. J. Mol. Biol. 2007, 367, 395)Part of HGF high affinity binding site Hepatocyte growth factor 90 kDb chain

Disulfide bonds

Biologically active MET activation, M


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