conversion of 1-boc-indoles to 1-boc-oxindoles

1
2004 Indole derivatives R 0140 Conversion of 1-Boc-indoles to 1-Boc-oxindoles. — Conversion of indoles to 2-(indolyl)borates and subsequent oxidation provides a general method for the synthe- sis of 2-oxindoles (II). — (VAZQUEZ, E.; PAYACK, J. F.; Tetrahedron Lett. 45 (2004) 35, 6549-6550; Dep. Process Res., Merck Res. Lab., Merck&Co., Inc., Rahway, NJ 07065, USA; Eng.) — Mais 49- 105

Upload: enrique-vazquez

Post on 06-Jun-2016

215 views

Category:

Documents


1 download

TRANSCRIPT

2004

Indole derivativesR 0140 Conversion of 1-Boc-indoles to 1-Boc-oxindoles. — Conversion of indoles to

2-(indolyl)borates and subsequent oxidation provides a general method for the synthe-sis of 2-oxindoles (II). — (VAZQUEZ, E.; PAYACK, J. F.; Tetrahedron Lett. 45 (2004) 35, 6549-6550; Dep. Process Res., Merck Res. Lab., Merck&Co., Inc., Rahway, NJ 07065, USA; Eng.) — Mais

49- 105